SCHEMBL30522720

SCHEMBL30522720

CC(C)(C)OC(=O)N1CCC2(CC1)CC2C(=O)Nc1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 12/20 0.56
GPR119 Q8TDV5 2/20 0.52
KEAP1 Q14145 1/20 0.51
NFE2L2 Q16236 1/20 0.51
JAK2 O60674 1/20 0.49
JAK1 P23458 1/20 0.49
CYP2C9 P11712 1/20 0.47
PTPN2 P17706 1/20 0.46
PTPN1 P18031 1/20 0.46
PTPN6 P29350 1/20 0.46
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24433501 1.00 NAMPT (0.56) NAMPTGPR119KEAP1NFE2L2JAK2
SCHEMBL24433521 0.87 PTPN2 (0.52) NAMPTGPR119KEAP1NFE2L2JAK2
SCHEMBL24442760 0.87 PTPN2 (0.49) NAMPTGPR119PTPN2PTPN1PTPN6
SCHEMBL24433507 0.83 JAK2 (0.49) NAMPTGPR119JAK2JAK1CYP2C9
SCHEMBL29657073 0.83 JAK2 (0.49) NAMPTGPR119JAK2JAK1CYP2C9
SCHEMBL24433402 0.83 JAK2 (0.51) NAMPTGPR119JAK2JAK1CYP2C9
SCHEMBL30522718 0.83 JAK2 (0.51) NAMPTGPR119JAK2JAK1CYP2C9
SCHEMBL24433406 0.83 MGLL (0.52)
SCHEMBL24433399 0.83 MGLL (0.52)
SCHEMBL24433407 0.83 MGLL (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116547274-A MAGL inhibitors H.隆德贝克有限公司 2023-08-04 CN disclosed