SCHEMBL30530286

SCHEMBL30530286

COc1cccc(C)c1NC(=O)c1ccc(Nc2ncc(SC)c(-c3cccnc3F)n2)cc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.43
PTK2 Q05397 9/20 0.42
AURKA O14965 2/20 0.42
AURKB Q96GD4 2/20 0.42
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PLK4 O00444 1/20 0.40
PDPK1 O15530 1/20 0.40
ABL1 P00519 1/20 0.40
EGFR P00533 1/20 0.40
ERBB2 P04626 1/20 0.40
NTRK1 P04629 1/20 0.40
GNAI2 P04899 1/20 0.40
LCK P06239 1/20 0.40
RET P07949 1/20 0.40
HCK P08631 1/20 0.40
ROS1 P08922 1/20 0.40
FGFR1 P11362 1/20 0.40
SRC P12931 1/20 0.40
GABRA1 P14867 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20187976 0.89 AURKA (0.45) AURKA
SCHEMBL30114850 0.89 AURKA (0.45) AURKA
SCHEMBL21799104 0.85 PTK2 (0.42) CHRNA7PTK2AURKAABL1
SCHEMBL30114830 0.85 PTK2 (0.42) CHRNA7PTK2AURKAABL1
SCHEMBL20188707 0.84 AURKA (0.47) PTK2AURKANTRK1KDRNTRK3
SCHEMBL20188270 0.81
SCHEMBL30114704 0.81
SCHEMBL20188131 0.79 PTK2 (0.44) PTK2AURKAABL1KDRLRRK2
SCHEMBL30530287 0.79 PTK2 (0.44) PTK2AURKAABL1KDRLRRK2
SCHEMBL20188007 0.77 AURKA (0.45) AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110139692-B Heteroaryl amine compounds for modulating hedgehog pathway and methods of making and using the same 财团法人生物技术开发中心 2023-08-25 CN claimed