SCHEMBL30530293

SCHEMBL30530293

CSc1cnc(Nc2ccc(C(=O)Nc3cc(CN4CCOCC4)ccc3C)cc2)cc1-c1ccc(F)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.53
NPC1 O15118 3/20 0.50
ACKR3 P25106 1/20 0.47
HTR2C P28335 2/20 0.46
MCHR1 Q99705 2/20 0.46
F10 P00742 1/20 0.45
WNT3A P56704 2/20 0.45
AURKA O14965 1/20 0.44
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
CDK2 P24941 1/20 0.44
AURKB Q96GD4 1/20 0.44
WDR5 P61964 2/20 0.44
ABL1 P00519 2/20 0.44
BCR P11274 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
GALR3 O60755 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21799076 1.00 RAB9A (0.53) RAB9ANPC1ACKR3HTR2CMCHR1
SCHEMBL20188084 0.92 ABL1 (0.49) ACKR3HTR2CMCHR1F10ABL1
SCHEMBL20188790 0.90 ABL1 (0.51) RAB9AABL1BCRSMN1; SMN2LMNA
SCHEMBL21799072 0.86 RAB9A (0.51) RAB9ANPC1ACKR3HTR2CMCHR1
SCHEMBL30530277 0.86 RAB9A (0.51) RAB9ANPC1ACKR3HTR2CMCHR1
SCHEMBL20188677 0.85 BRAF (0.49) ABL1BCRLMNAMAPK14
SCHEMBL21799087 0.83 ABL1 (0.47) ABL1BCRLMNAMAPK14
SCHEMBL30114739 0.83 ABL1 (0.47) ABL1BCRLMNAMAPK14
SCHEMBL21799112 0.81 RAB9A (0.49) RAB9AABL1BCRLMNAMAPK14
SCHEMBL30114702 0.81 RAB9A (0.49) RAB9AABL1BCRLMNAMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110139692-B Heteroaryl amine compounds for modulating hedgehog pathway and methods of making and using the same 财团法人生物技术开发中心 2023-08-25 CN claimed
CN-110139692-B Heteroaryl amine compounds for modulating hedgehog pathway and methods of making and using the same 财团法人生物技术开发中心 2023-08-25 CN disclosed