SCHEMBL30540451

SCHEMBL30540451

CC1(C)CCc2c(C=O)cc(C(N)=O)nc21

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EEF2K O00418 18/20 0.42
GRM2 Q14416 1/20 0.39
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30540646 0.84 MAPK1 (0.34) EEF2K
SCHEMBL30540577 0.78 EEF2K (0.38) EEF2KGRM2LMNA
SCHEMBL30540558 0.74 GRM2 (0.37) GRM2LMNA
SCHEMBL30625623 0.73 EEF2K (0.35) EEF2KGRM2LMNA
SCHEMBL30625415 0.72 MAPK1 (0.33)
SCHEMBL30625588 0.70 EEF2K (0.36) EEF2K
SCHEMBL30540659 0.70 EEF2K (0.36) EEF2KLMNA
SCHEMBL30625617 0.70 EEF2K (0.37) EEF2KGRM2
SCHEMBL31115335 0.69 ERN1 (0.34) GRM2LMNA
SCHEMBL30540572 0.69 ERN1 (0.34) GRM2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4476219-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BeiGene, Ltd. (KY) 2024-12-18 EP disclosed
CN-118696043-A Heterocyclic compounds, compositions thereof and methods of treatment therewith 百济神州有限公司 2024-09-24 CN disclosed
WO-2023151642-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BEIGENE , LTD. (KY) 2023-08-17 WO disclosed
WO-2023151636-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BEIGENE , LTD. (KY) 2023-08-17 WO disclosed