SCHEMBL30544071

SCHEMBL30544071

N[C@@H](Cc1c(F)ccc(F)c1F)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 3/20 0.48
PKM P14618 2/20 0.48
PTGS1 P23219 2/20 0.48
ALPI P09923 1/20 0.48
XIAP P98170 1/20 0.48
USP2 O75604 3/20 0.44
HSD17B10 Q99714 3/20 0.44
ALOX15 P16050 2/20 0.44
HIF1A Q16665 2/20 0.44
KDM4E B2RXH2 2/20 0.44
RECQL P46063 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
TNF P01375 1/20 0.44
RGS12 O14924 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
NFKB1 P19838 1/20 0.44
CASP1 P29466 1/20 0.44
BRCA1 P38398 1/20 0.44
THPO P40225 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3624208 0.86 SLC7A5 (0.43) SLC7A5PKMPTGS1ALPIXIAP
SCHEMBL188587 0.83 SLC7A5 (0.55) SLC7A5PKMPTGS1ALPIXIAP
SCHEMBL20514005 0.83 SLC7A5 (0.55) SLC7A5PKMPTGS1ALPIXIAP
SCHEMBL188588 0.83 SLC7A5 (0.55) SLC7A5PKMPTGS1ALPIXIAP
SCHEMBL7280604 0.83 USP2 (0.50) SLC7A5PKMPTGS1ALPIXIAP
SCHEMBL5285947 0.83 USP2 (0.50) SLC7A5PKMPTGS1ALPIXIAP
SCHEMBL11434038 0.81 SLC7A5 (0.50) SLC7A5PKMPTGS1ALPIXIAP
SCHEMBL1527383 0.80 USP2 (0.51) SLC7A5PKMPTGS1ALPIXIAP
SCHEMBL1516481 0.80 USP2 (0.47) SLC7A5PKMPTGS1ALPIXIAP
SCHEMBL13957611 0.80 USP2 (0.47) SLC7A5PKMPTGS1ALPIXIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250179465-A1 SITE-SPECIFIC ENCODING OF FLUORINATED PHENYLALANINE RESIDUES IN BACTERIAL AND MAMMALIAN CELLS UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2025-06-05 US claimed
EP-4479526-A1 SITE-SPECIFIC ENCODING OF FLUORINATED PHENYLALANINE RESIDUES IN BACTERIAL AND MAMMALIAN CELLS University of Iowa Research Foundation (US) 2024-12-25 EP claimed
WO-2023158761-A1 SITE-SPECIFIC ENCODING OF FLUORINATED PHENYLALANINE RESIDUES IN BACTERIAL AND MAMMALIAN CELLS UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2023-08-24 WO claimed
US-20250179465-A1 SITE-SPECIFIC ENCODING OF FLUORINATED PHENYLALANINE RESIDUES IN BACTERIAL AND MAMMALIAN CELLS UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2025-06-05 US disclosed
EP-4479526-A1 SITE-SPECIFIC ENCODING OF FLUORINATED PHENYLALANINE RESIDUES IN BACTERIAL AND MAMMALIAN CELLS University of Iowa Research Foundation (US) 2024-12-25 EP disclosed
WO-2023158761-A1 SITE-SPECIFIC ENCODING OF FLUORINATED PHENYLALANINE RESIDUES IN BACTERIAL AND MAMMALIAN CELLS UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2023-08-24 WO disclosed