SCHEMBL30547271

SCHEMBL30547271

COC(=O)C(Cc1cccnc1)NC(=O)OC(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.55
NLRP3 Q96P20 1/20 0.54
CYP3A4 P08684 8/20 0.52
SCN9A Q15858 1/20 0.51
CTSS P25774 3/20 0.50
CTSB P07858 3/20 0.50
CTSL P07711 2/20 0.50
CTSK P43235 2/20 0.50
ACE P12821 1/20 0.48
REN P00797 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21875889 1.00 KLK5 (0.55) KLK5NLRP3CYP3A4SCN9ACTSS
SCHEMBL12290542 1.00 KLK5 (0.55) KLK5NLRP3CYP3A4SCN9ACTSS
SCHEMBL2367394 1.00 KLK5 (0.55) KLK5NLRP3CYP3A4SCN9ACTSS
SCHEMBL29588090 0.94 CYP3A4 (0.52) KLK5NLRP3CYP3A4SCN9ACTSS
SCHEMBL8125933 0.94 CYP3A4 (0.52) KLK5NLRP3CYP3A4SCN9ACTSS
SCHEMBL3820580 0.92 KLK5 (0.48) KLK5NLRP3CYP3A4SCN9ACTSS
SCHEMBL2367071 0.91 KLK5 (0.48) KLK5NLRP3CYP3A4SCN9ACTSS
SCHEMBL27683505 0.91 KLK5 (0.48) KLK5NLRP3CYP3A4SCN9ACTSS
SCHEMBL13323781 0.91 KLK5 (0.48) KLK5NLRP3CYP3A4SCN9ACTSS
SCHEMBL479037 0.89 ACE (0.61) CYP3A4SCN9ACTSSCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116496255-A NLRP3 inhibitors 杭州邦顺制药有限公司 2023-07-28 CN disclosed