SCHEMBL30558136

SCHEMBL30558136

COc1ccc(F)cc1C(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSS P25774 3/20 0.41
CTSK P43235 3/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 2/20 0.39
GAA P10253 1/20 0.39
AAK1 Q2M2I8 1/20 0.39
TRPA1 O75762 1/20 0.38
LMNA P02545 2/20 0.37
CTSA P10619 2/20 0.37
ITGA4 P13612 1/20 0.37
ITGB7 P26010 1/20 0.37
ACE P12821 1/20 0.37
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
S1PR3 Q99500 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29364123 1.00 CTSS (0.41) CTSSCTSKKDM4EALDH1A1GAA
SCHEMBL3815433 1.00 CTSS (0.41) CTSSCTSKKDM4EALDH1A1GAA
SCHEMBL3762203 0.86 CTSS (0.43) CTSSCTSKALDH1A1AAK1TRPA1
SCHEMBL30765251 0.86 CTSS (0.43) CTSSCTSKALDH1A1AAK1TRPA1
SCHEMBL17395943 0.85 CTSS (0.49) CTSSCTSKITGA4ITGB7ACE
SCHEMBL21777294 0.85 CTSS (0.49) CTSSCTSKITGA4ITGB7ACE
SCHEMBL265969 0.85 CTSS (0.49) CTSSCTSKITGA4ITGB7ACE
SCHEMBL23414163 0.84 CTSS (0.40) CTSSCTSKKDM4EALDH1A1GAA
SCHEMBL3822263 0.83 CTSS (0.43) CTSSCTSKAAK1TRPA1ACE
SCHEMBL29571131 0.83 CTSS (0.43) CTSSCTSKAAK1TRPA1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116693518-A Synthesis and application of EGFR inhibitor 江南大学 2023-09-05 CN disclosed