SCHEMBL30559705

SCHEMBL30559705

COc1cc(C(C)(F)F)nc(N)n1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
RAB9A P51151 1/20 0.45
HSD17B10 Q99714 2/20 0.44
KDM4E B2RXH2 5/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
NUDT1 P36639 3/20 0.41
GRM4 Q14833 1/20 0.41
GAA P10253 2/20 0.38
AURKA O14965 1/20 0.36
PDPK1 O15530 1/20 0.36
TGFBR1 P36897 1/20 0.36
ROCK1 Q13464 1/20 0.36
AURKB Q96GD4 1/20 0.36
MAPT P10636 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26978084 1.00 NPC1 (0.45) NPC1ALDH1A1RAB9AHSD17B10KDM4E
SCHEMBL5891451 0.87 HSP90AA1 (0.58) NPC1ALDH1A1RAB9AHSD17B10KDM4E
SCHEMBL24714024 0.85 HSD17B10 (0.61) NPC1ALDH1A1RAB9AHSD17B10KDM4E
SCHEMBL31543553 0.78 ALDH1A1 (0.40) ALDH1A1KDM4EGAAMAPTCYP1A2
SCHEMBL26685699 0.78 ALDH1A1 (0.40) ALDH1A1KDM4EGAAMAPTCYP1A2
SCHEMBL151590 0.77 ALDH1A1 (0.59) NPC1ALDH1A1RAB9AHSD17B10KDM4E
SCHEMBL7804008 0.76 NPC1 (0.46) NPC1ALDH1A1RAB9AHSD17B10KDM4E
Hydrochloric Acid SCHEMBL10746200 0.75 ALDH1A1 (0.57) NPC1ALDH1A1RAB9AHSD17B10KDM4E
SCHEMBL10645339 0.74 NPC1 (0.45) NPC1ALDH1A1RAB9AHSD17B10KDM4E
SCHEMBL31581577 0.74 GAA (0.35) NPC1ALDH1A1RAB9AKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116829550-A Pyrimidine-2-ylsulfonamide derivatives 豪夫迈·罗氏有限公司 2023-09-29 CN disclosed