SCHEMBL30560100

SCHEMBL30560100

CCOC(=O)/C=C/c1cnc(SC)nc1NC1CCCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
MAPT P10636 3/20 0.41
NR2F2 P24468 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
MAPK1 P28482 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
TDP1 Q9NUW8 2/20 0.40
GABBR2 O75899 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
GABBR1 Q9UBS5 1/20 0.40
LMNA P02545 3/20 0.40
SYK P43405 2/20 0.40
NPC1 O15118 1/20 0.40
S1PR2 O95136 1/20 0.40
XBP1 P17861 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4715488 1.00 ALDH1A1 (0.41) ALDH1A1MAPTNR2F2NPSR1MAPK1
SCHEMBL30498445 1.00 ALDH1A1 (0.41) ALDH1A1MAPTNR2F2NPSR1MAPK1
SCHEMBL16094578 1.00 ALDH1A1 (0.41) ALDH1A1MAPTNR2F2NPSR1MAPK1
SCHEMBL4716299 0.99 MEN1 (0.41) ALDH1A1MAPTNR2F2NPSR1MAPK1
SCHEMBL4760645 0.99 MEN1 (0.41) ALDH1A1MAPTNR2F2NPSR1MAPK1
SCHEMBL4711389 0.96 ALDH1A1 (0.43) ALDH1A1MAPTNR2F2NPSR1MAPK1
SCHEMBL4715139 0.96 ALDH1A1 (0.43) ALDH1A1MAPTNR2F2NPSR1MAPK1
SCHEMBL14914394 0.89 KMT2A (0.43) ALDH1A1KDM4EMEN1KMT2ATDP1
SCHEMBL30872620 0.89 KMT2A (0.43) ALDH1A1KDM4EMEN1KMT2ATDP1
SCHEMBL14914395 0.89 KMT2A (0.43) ALDH1A1KDM4EMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3733184-B1 PYRIMIDINE COMPOUNDS FOR USE IN THE TREATMENT OF CANCER ICAHN SCHOOL MED MOUNT SINAI (US) 2023-08-30 EP disclosed