SCHEMBL30573103

SCHEMBL30573103

COC(=O)c1cncc(Br)c1N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.49
ALDH1A1 P00352 5/20 0.49
GAA P10253 5/20 0.49
GLA P06280 3/20 0.49
TSHR P16473 2/20 0.46
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
CYP2C9 P11712 1/20 0.43
HSD17B10 Q99714 5/20 0.42
CFTR P13569 1/20 0.42
CYP3A4 P08684 1/20 0.40
PKM P14618 1/20 0.40
POLB P06746 1/20 0.40
MAPK1 P28482 1/20 0.40
ATM Q13315 2/20 0.40
HPGD P15428 3/20 0.39
CASP1 P29466 2/20 0.39
CASP7 P55210 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17603665 1.00 KDM4E (0.49) KDM4EALDH1A1GAAGLATSHR
SCHEMBL17802090 0.81 ALDH1A1 (0.43) KDM4EALDH1A1GAAGLATSHR
SCHEMBL16694522 0.80 GAA (0.42) KDM4EALDH1A1GAAGLATSHR
SCHEMBL31184958 0.80 ATM (0.44) KDM4EALDH1A1GAAGLATSHR
SCHEMBL21750020 0.80 ATM (0.44) KDM4EALDH1A1GAAGLATSHR
SCHEMBL9939057 0.80 ATM (0.44) KDM4EALDH1A1GAAGLATSHR
SCHEMBL30573060 0.80 KDM4E (0.50) KDM4EALDH1A1GAAGLATSHR
SCHEMBL2003190 0.80 KDM4E (0.50) KDM4EALDH1A1GAAGLATSHR
SCHEMBL17619233 0.79 SMN1; SMN2 (0.33) KDM4EALDH1A1GAAGLAKMT2A
SCHEMBL16694957 0.79 SOS1 (0.44) KDM4EALDH1A1GAAGLATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4511114-A1 HETEROARYL COMPOUNDS FOR THE TREATMENT OF PAIN Vertex Pharmaceuticals Incorporated (US) 2025-02-26 EP disclosed
WO-2023205778-A1 HETEROARYL COMPOUNDS FOR THE TREATMENT OF PAIN VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-10-26 WO disclosed