SCHEMBL30587486

SCHEMBL30587486

COC(=O)c1ncc2c(n1)C1(CCOCC1)OC2

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.32
HPGD P15428 2/20 0.32
ALOX15 P16050 1/20 0.32
MGLL Q99685 1/20 0.32
HSD17B10 Q99714 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MAPK1 P28482 1/20 0.31
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
MEN1 O00255 1/20 0.30
APAF1 O14727 1/20 0.30
TDP2 O95551 1/20 0.30
NSD2 O96028 1/20 0.30
PLA2G1B P04054 1/20 0.30
HSP90AA1 P07900 1/20 0.30
PLCG1 P19174 1/20 0.30
GALK1 P51570 1/20 0.30
BLM P54132 1/20 0.30
KMT2A Q03164 1/20 0.30
PDIA6 Q15084 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18366858 1.00 ALDH1A1 (0.32) ALDH1A1HPGDALOX15MGLLHSD17B10
SCHEMBL18366850 0.93
SCHEMBL30587509 0.90 NPC1 (0.31) ALDH1A1HPGDNPC1RAB9AKMT2A
SCHEMBL18367169 0.90 NPC1 (0.31) ALDH1A1HPGDNPC1RAB9AKMT2A
SCHEMBL18366791 0.90 NPC1 (0.31) ALDH1A1HPGDNPC1RAB9AKMT2A
SCHEMBL30587561 0.90 NPC1 (0.31) ALDH1A1HPGDNPC1RAB9AKMT2A
SCHEMBL30587621 0.86
SCHEMBL18366945 0.86
SCHEMBL18366859 0.84 POLB (0.33)
SCHEMBL19658801 0.83 KDM4E (0.36) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111269221-B Bicyclic lactams and methods of use thereof 豪夫迈·罗氏有限公司 2023-09-26 CN disclosed