SCHEMBL30593161

SCHEMBL30593161

CCOC(=O)c1c(C)nc(O)c([N+](=O)[O-])c1O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.45
POLB P06746 2/20 0.43
ADORA3 P0DMS8 2/20 0.42
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 3/20 0.41
RAB9A P51151 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
LMNA P02545 2/20 0.41
GAA P10253 2/20 0.41
NPC1 O15118 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PDE4D Q08499 2/20 0.41
TP53 P04637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
RECQL P46063 1/20 0.40
PKM P14618 1/20 0.40
HTT P42858 1/20 0.40
PDE4B Q07343 1/20 0.39
CA12 O43570 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11626481 1.00 MAPT (0.45) MAPTPOLBADORA3ALDH1A1KDM4E
SCHEMBL2574309 0.82 MAPT (0.41) MAPTPOLBALDH1A1KDM4ENPSR1
SCHEMBL11614853 0.80 TDP1 (0.39) MAPTPOLBALDH1A1RAB9ASMN1; SMN2
SCHEMBL31336329 0.78 ADORA3 (0.48) MAPTPOLBADORA3ALDH1A1KDM4E
SCHEMBL26608431 0.78 ADORA3 (0.48) MAPTPOLBADORA3ALDH1A1KDM4E
SCHEMBL30593158 0.75 POLB (0.42) MAPTPOLBADORA3ALDH1A1KDM4E
SCHEMBL11628165 0.75 POLB (0.42) MAPTPOLBADORA3ALDH1A1KDM4E
SCHEMBL14183027 0.75 ADORA3 (0.50) MAPTPOLBADORA3ALDH1A1KDM4E
SCHEMBL9270724 0.73 POLB (0.47) MAPTPOLBADORA3ALDH1A1KDM4E
SCHEMBL11728849 0.73 KDM4E (0.46) MAPTPOLBALDH1A1KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4511115-A1 HETEROARYL COMPOUNDS FOR THE TREATMENT OF PAIN Vertex Pharmaceuticals Incorporated (US) 2025-02-26 EP disclosed
WO-2023205468-A1 HETEROARYL COMPOUNDS FOR THE TREATMENT OF PAIN VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-10-26 WO disclosed