SCHEMBL30593231

SCHEMBL30593231

CC(C)(C)OC(=O)N1CCc2cc(-c3coc4ccccc34)ccc2C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.56
NR1H2 P55055 1/20 0.50
NAMPT P43490 4/20 0.44
MAPK1 P28482 2/20 0.43
ALDH2 P05091 2/20 0.40
UCHL1 P09936 1/20 0.39
PRMT5 O14744 1/20 0.39
WDR77 Q9BQA1 1/20 0.39
NPC1 O15118 1/20 0.39
PIK3CA P42336 1/20 0.39
MTOR P42345 1/20 0.39
KDM4E B2RXH2 2/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29084888 1.00 ESR2 (0.56) ESR2NR1H2NAMPTMAPK1ALDH2
SCHEMBL31070534 0.92 HDAC1 (0.44) ESR2NR1H2NAMPTMAPK1ALDH2
SCHEMBL30593261 0.82 ESR2 (0.60) ESR2NR1H2NAMPTMAPK1UCHL1
SCHEMBL25407478 0.82 ESR2 (0.60) ESR2NR1H2NAMPTMAPK1UCHL1
SCHEMBL30593270 0.81 ESR2 (0.69) ESR2NR1H2NAMPTMAPK1UCHL1
SCHEMBL23124526 0.81 ESR2 (0.69) ESR2NR1H2NAMPTMAPK1UCHL1
SCHEMBL31428709 0.78 ESR2 (0.54) ESR2NR1H2NAMPTMAPK1KDM4E
SCHEMBL24842903 0.78 ESR2 (0.65) ESR2NR1H2NAMPTMAPK1UCHL1
SCHEMBL22821172 0.77 ESR2 (0.57) ESR2NR1H2NAMPTMAPK1UCHL1
SCHEMBL25405200 0.77 ESR2 (0.63) ESR2NR1H2NAMPTMAPK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118742543-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2024-10-01 CN disclosed
CN-116789641-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2023-09-22 CN disclosed