SCHEMBL30593261

SCHEMBL30593261

CC(C)(C)OC(=O)N1CCc2cc(-c3cccc4ccccc34)ccc2C1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.60
NR1H2 P55055 1/20 0.53
NAMPT P43490 1/20 0.46
UCHL1 P09936 1/20 0.45
MAPK1 P28482 1/20 0.45
TMPRSS2 O15393 1/20 0.42
KDM4E B2RXH2 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
JAK2 O60674 3/20 0.42
JAK3 P52333 3/20 0.42
PTK2 Q05397 3/20 0.42
PDK4 Q16654 1/20 0.42
PARP1 P09874 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41
PARP2 Q9UGN5 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
PPARG P37231 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25407478 1.00 ESR2 (0.60) ESR2NR1H2NAMPTUCHL1MAPK1
SCHEMBL24842903 0.85 ESR2 (0.65) ESR2NR1H2NAMPTUCHL1MAPK1
SCHEMBL22821172 0.83 ESR2 (0.57) ESR2NR1H2NAMPTUCHL1MAPK1
SCHEMBL30593270 0.83 ESR2 (0.69) ESR2NR1H2NAMPTUCHL1MAPK1
SCHEMBL23124526 0.83 ESR2 (0.69) ESR2NR1H2NAMPTUCHL1MAPK1
SCHEMBL31428709 0.83 ESR2 (0.54) ESR2NR1H2NAMPTMAPK1KDM4E
SCHEMBL29084888 0.82 ESR2 (0.56) ESR2NR1H2NAMPTUCHL1MAPK1
SCHEMBL30593231 0.82 ESR2 (0.56) ESR2NR1H2NAMPTUCHL1MAPK1
SCHEMBL22821061 0.82 ESR2 (0.58) ESR2NR1H2NAMPTUCHL1MAPK1
SCHEMBL29733605 0.82 ESR2 (0.58) ESR2NR1H2NAMPTUCHL1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118742543-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2024-10-01 CN disclosed
CN-116789641-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2023-09-22 CN disclosed