SCHEMBL30595387

SCHEMBL30595387

CCCCCC(CC)c1cccc2onc(N)c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.40
FLT3 P36888 9/20 0.40
KIT P10721 8/20 0.40
AURKB Q96GD4 7/20 0.40
MET P08581 3/20 0.40
MAP4K4 O95819 2/20 0.40
PDGFRB P09619 2/20 0.40
PIM1 P11309 2/20 0.40
FGFR1 P11362 2/20 0.40
PDGFRA P16234 2/20 0.40
PRKACA P17612 2/20 0.40
LTK P29376 2/20 0.40
GRK5 P34947 2/20 0.40
CDK8 P49336 2/20 0.40
CDK7 P50613 2/20 0.40
CDK9 P50750 2/20 0.40
LIMK1 P53667 2/20 0.40
MAP2K1 Q02750 2/20 0.40
ACVR1 Q04771 2/20 0.40
MST1R Q04912 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30595391 0.83 KDR (0.32) KDRFLT3KITAURKBMET
SCHEMBL22304364 0.75 KDR (0.50) KDRFLT3KITAURKBMET
SCHEMBL8524531 0.72 NR1I2 (0.45) NR1I2
SCHEMBL29814520 0.71 ADA (0.39) FAAHDHFRNR1I2
SCHEMBL29745185 0.71 NR1I2 (0.40) NR1I2
SCHEMBL29744995 0.70 NR1I2 (0.42) DHFRNR1I2
SCHEMBL7104911 0.70 NR1I2 (0.42) DHFRNR1I2
SCHEMBL10633096 0.70 NR1I2 (0.42) DHFRNR1I2
SCHEMBL19695714 0.68 KDR (0.50) KDRFLT3KITAURKBMET
SCHEMBL29814823 0.68 NOS2 (0.39) DHFREGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116804005-A Kinesin KIF18A inhibitor and application thereof 上海湃隆生物科技有限公司 2023-09-26 CN disclosed