SCHEMBL305967

SCHEMBL305967

CN1CCNc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRPF1 P55201 1/20 0.47
BRD4 O60885 2/20 0.44
AVPR1A P37288 2/20 0.43
PIM1 P11309 1/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
GAA P10253 2/20 0.40
ADRB1 P08588 3/20 0.37
HSD17B3 P37058 1/20 0.37
CREBBP Q92793 1/20 0.36
MAPK1 P28482 1/20 0.36
ALDH1A1 P00352 1/20 0.34
HTR3E A5X5Y0 1/20 0.34
HTR3B O95264 1/20 0.34
DRD2 P14416 1/20 0.34
CYP2C19 P33261 1/20 0.34
DRD3 P35462 1/20 0.34
HTR3A P46098 1/20 0.34
HTR6 P50406 1/20 0.34
HTR3D Q70Z44 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30463209 1.00 BRPF1 (0.47) BRPF1BRD4AVPR1APIM1MEN1
Hydrochloric Acid SCHEMBL23882148 0.98 BRPF1 (0.46) BRPF1BRD4AVPR1APIM1MEN1
SCHEMBL2631721 0.88 MEN1 (0.46) BRPF1BRD4AVPR1APIM1MEN1
SCHEMBL12387711 0.83 BRPF1 (0.41) BRPF1BRD4AVPR1APIM1MEN1
SCHEMBL30738818 0.78 BRPF1 (0.50) BRPF1BRD4AVPR1AMEN1KMT2A
SCHEMBL4013751 0.78 BRPF1 (0.50) BRPF1BRD4AVPR1AMEN1KMT2A
SCHEMBL30379824 0.77 KDM4E (0.54) BRD4MEN1KMT2AGAAALDH1A1
SCHEMBL28833094 0.77 BRD4 (0.41) BRPF1BRD4AVPR1APIM1MEN1
SCHEMBL14497763 0.76 MEN1 (0.49) BRPF1BRD4AVPR1APIM1MEN1
SCHEMBL3311949 0.75 AVPR1A (0.40) BRPF1BRD4AVPR1APIM1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 141 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116199675-A Rhodamine fluorescence quenching agent and synthesis and application thereof 中国科学院大连化学物理研究所 2023-06-02 CN claimed
WO-1999065865-A1 NOVEL 3,4-DIAMINOPHENOL DERIVATIVES AND THEIR USE HANS SCHWARZKOPF GMBH & CO. KG (DE) 1999-12-23 WO claimed
WO-1999065891-A1 NOVEL 2,4-DIAMINOPHENOL DERIVATIVES AND THE USE THEREOF HANS SCHWARZKOPF GMBH & CO. KG (DE) 1999-12-23 WO claimed
EP-0257583-B1 PROCESS FOR ORTHO-CYANATION OF PHENOLS OR PHENYLAMINES SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1992-01-08 EP claimed
EP-0266849-B1 PROCESS FOR INTRODUCING A THIOCARBOXYLIC ESTER GROUP AT THE ORTHO-POSITION OF PHENOLS OR PHENYLAMINES SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1991-03-13 EP claimed
US-4857645-A Process for introducing a thiocarboxylic ester group at the orthoposition of phenols or phenylamines SHIONOGI & CO., LTD. (JP) 1989-08-15 US claimed
US-4774331-A THIOCYANATION IN PRESENCE OF BORON TRIFLUORIDE SHIONOGI & CO., LTD. (JP) 1988-09-27 US claimed
EP-0266849-A1 Process for introducing a thiocarboxylic ester group at the ortho-position of phenols or phenylamines SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1988-05-11 EP claimed
EP-0257583-A1 Process for ortho-cyanation of phenols or phenylamines SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1988-03-02 EP claimed
US-20250171420-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME MONTE ROSA THERAPEUTICS AG (CH) 2025-05-29 US disclosed
EP-4540240-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME Monte Rosa Therapeutics AG (CH) 2025-04-23 EP disclosed
WO-2024123991-A1 TREATMENT OF AUTOIMMUNE AND INFLAMMATORY DISORDERS WITH INHIBITORS OF BET FAMILY BDII BROMODOMAIN POSEIDON INNOVATION 1, INC. (US) 2024-06-13 WO disclosed
WO-2024123999-A1 TREATMENT OF GRAFT-VERSUS-HOST DISEASE WITH INHIBITORS OF BET FAMILY BDII BROMODOMAIN POSEIDON INNOVATION 1, INC. (US) 2024-06-13 WO disclosed
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
WO-1999065891-A1 NOVEL 2,4-DIAMINOPHENOL DERIVATIVES AND THE USE THEREOF HANS SCHWARZKOPF GMBH & CO. KG (DE) 1999-12-23 WO disclosed
US-5459142-A Autoimmune disease, atherosclerosis, antiischemic agents and nephritis OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-10-17 US disclosed
US-5322842-A Tricyclic benzodiazepine derivates, their preparation, and pharmaceutical compositions containing them FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-06-21 US disclosed
EP-0544909-A1 TRICYCLIC BENZODIAZEPINE DERIVATES THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-06-09 EP disclosed
WO-1992003438-A1 TRICYCLIC BENZODIAZEPINE DERIVATES THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-03-05 WO disclosed
US-4576954-A Anti-rheumatic 5-(substituted amino)-1,2-dithiol-3-one compounds and their use PHONE-POULENC SANTE (FR) 1986-03-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250171420-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME PSMA1, CSNK1G1, CSNK1A1 BRPF1 2325/4885BRD4 611/4885AVPR1A 4207/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.