SCHEMBL30599698

SCHEMBL30599698

COC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(NC(=O)Nc2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 7/20 0.71
HCRTR2 O43614 7/20 0.71
BRD4 O60885 5/20 0.66
POLB P06746 2/20 0.61
BRD2 P25440 4/20 0.57
HTT P42858 5/20 0.54
MAPT P10636 4/20 0.54
XBP1 P17861 2/20 0.54
MEN1 O00255 2/20 0.53
LMNA P02545 2/20 0.53
TP53 P04637 2/20 0.53
KMT2A Q03164 2/20 0.53
ALOX15 P16050 1/20 0.53
MAPK1 P28482 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.52
NPSR1 Q6W5P4 2/20 0.52
ALOX12 P18054 1/20 0.52
BRD3 Q15059 3/20 0.52
BRDT Q58F21 3/20 0.52
CYP3A4 P08684 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20291205 1.00 HCRTR1 (0.71) HCRTR1HCRTR2BRD4POLBBRD2
SCHEMBL20291072 0.90 BRD4 (0.73) HCRTR1HCRTR2BRD4POLBBRD2
SCHEMBL23787106 0.89 BRD4 (0.72) HCRTR1HCRTR2BRD4POLBBRD2
SCHEMBL20291414 0.86 BRD4 (0.66) HCRTR1HCRTR2BRD4HTTMAPT
SCHEMBL20291227 0.85 HCRTR1 (0.55) HCRTR1HCRTR2BRD4BRD2MAPK1
SCHEMBL20291395 0.84 HCRTR1 (0.56) HCRTR1HCRTR2BRD4BRD2MAPT
SCHEMBL20291390 0.83 ALDH1A1 (0.65) HCRTR1HCRTR2BRD4HTTMAPT
SCHEMBL20291277 0.83 BRD4 (0.57) HCRTR1HCRTR2BRD4BRD2KMT2A
SCHEMBL20291003 0.83 BRD4 (0.60) HCRTR1HCRTR2BRD4POLBBRD2
SCHEMBL30599699 0.83 BRD4 (0.60) HCRTR1HCRTR2BRD4POLBBRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3554503-B1 INHIBITORS OF BROMODOMAIN-CONTAINING PROTEIN 4 (BRD4) UNIV TEXAS (US) 2023-10-04 EP disclosed