SCHEMBL30610258

SCHEMBL30610258

CCc1nccnc1CC(C)C

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 3/20 0.40
PDE3A Q14432 3/20 0.40
KDM4E B2RXH2 1/20 0.39
USP2 O75604 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TRPM8 Q7Z2W7 1/20 0.35
GCK P35557 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13980103 1.00 PDE3B (0.40) PDE3BPDE3AKDM4EUSP2HPGD
SCHEMBL18858530 0.90 PDE3B (0.44) PDE3BPDE3AKDM4EUSP2HPGD
SCHEMBL27355631 0.83
SCHEMBL24202601 0.82 PDE3B (0.30) PDE3BPDE3A
SCHEMBL27289776 0.82 PDE3B (0.30) PDE3BPDE3A
SCHEMBL34472956 0.82 PDE3B (0.39) PDE3BPDE3A
SCHEMBL1131513 0.82 PDE3B (0.39) PDE3BPDE3A
Ammonia Solution, Strong SCHEMBL28980458 0.79 PDE3B (0.38) PDE3BPDE3A
SCHEMBL30110738 0.76 PDE3B (0.40) PDE3BPDE3AKDM4EUSP2HPGD
SCHEMBL1532455 0.76 PDE3B (0.40) PDE3BPDE3AKDM4EUSP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11945785-B2 Pyrazine compounds as inhibitors of FLT3 BIOMEA FUSION, INC. (US) 2024-04-02 US disclosed
US-20230339867-A1 PYRAZINE COMPOUNDS AS INHIBITORS OF FLT3 BIOMEA FUSION, INC. 2023-10-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11945785-B2 Pyrazine compounds as inhibitors of FLT3 FLT3, MCL1, JAK2 PDE3B 2138/4885PDE3A 2063/4885KDM4E 2031/4885
US-20230339867-A1 PYRAZINE COMPOUNDS AS INHIBITORS OF FLT3 FLT3, MCL1, CSF3R PDE3B 2642/4885PDE3A 2513/4885KDM4E 2175/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.