SCHEMBL30615331

SCHEMBL30615331

O=c1[nH]c2ncccc2n1-c1cnc2ccccc2c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.47
PRKCQ Q04759 12/20 0.46
PDE2A O00408 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
PRKCA P17252 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
HTR3A P46098 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
CYP2A6 P11509 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21463917 1.00 DAO (0.47) DAOPRKCQPDE2APDE3BPDE3A
SCHEMBL21463768 0.87 PRKCQ (0.50) DAOPRKCQPRKCAALDH1A1
SCHEMBL30615354 0.87 PRKCQ (0.50) DAOPRKCQPRKCAALDH1A1
SCHEMBL30615630 0.83 AURKA (0.56)
SCHEMBL11511885 0.79 DAO (0.58) DAOPRKCQPRKCAALDH1A1
SCHEMBL30794441 0.77 DAO (0.53) DAOPRKCQPRKCAALDH1A1
SCHEMBL30257859 0.76 DAO (0.55) DAOPRKCQPRKCAALDH1A1
SCHEMBL21463351 0.75 GABRP (0.51) ALDH1A1
SCHEMBL30615474 0.75 GABRP (0.51) ALDH1A1
SCHEMBL30615505 0.75 AURKA (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111868037-B Fused cyclic urea derivatives as CRHR2 antagonists 拉夸里亚创药株式会社 2023-10-13 CN disclosed