SCHEMBL30620596

SCHEMBL30620596

O=C(O)c1ccccc1-c1ccccn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.52
TDP1 Q9NUW8 1/20 0.52
KDM4C Q9H3R0 2/20 0.51
KDM6B O15054 1/20 0.51
KDM4A O75164 1/20 0.51
KDM5C P41229 1/20 0.51
KDM2A Q9Y2K7 1/20 0.51
KDM3A Q9Y4C1 1/20 0.51
L3MBTL1 Q9Y468 3/20 0.50
ALDH1A1 P00352 2/20 0.50
ALOX15 P16050 2/20 0.50
BLM P54132 2/20 0.50
CYP3A4 P08684 1/20 0.50
MAPT P10636 1/20 0.50
TSHR P16473 1/20 0.50
AGER Q15109 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
GRM5 P41594 1/20 0.50
DHODH Q02127 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1173966 1.00 KDM4E (0.52) KDM4ETDP1KDM4CKDM6BKDM4A
Trifluoroacetic Acid SCHEMBL29693948 0.90 KDM4E (0.46) KDM4ETDP1KDM4CKDM6BKDM4A
SCHEMBL9202323 0.86 KDM4E (0.50) KDM4ETDP1KDM4CKDM6BKDM4A
SCHEMBL9235039 0.86 HNF4A (0.59) KDM4ETDP1KDM4CKDM6BKDM4A
SCHEMBL28459406 0.86 GRM5 (0.49) KDM4ETDP1KDM4CKDM6BKDM4A
SCHEMBL31575871 0.85 KMT2A (0.55) KDM4ETDP1KDM4CKDM6BKDM4A
SCHEMBL27591915 0.85 KMT2A (0.55) KDM4ETDP1KDM4CKDM6BKDM4A
SCHEMBL17427074 0.85 KDM4E (0.56) KDM4ETDP1KDM4CKDM6BKDM4A
SCHEMBL3555744 0.84 NAPRT (0.50) KDM4ETDP1KDM4CKDM6BKDM4A
SCHEMBL31317750 0.84 KDM4E (0.68) KDM4ETDP1KDM4CKDM6BKDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116601131-A CTPS1 inhibitor and application thereof 林伯士克洛索有限公司 2023-08-15 CN disclosed