SCHEMBL30622249

SCHEMBL30622249

COCc1c(Br)cccc1-c1nnc(C)o1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.47
NPC1 O15118 8/20 0.41
RAB9A P51151 8/20 0.41
TDP1 Q9NUW8 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 6/20 0.38
ALDH1A1 P00352 5/20 0.38
HPGD P15428 4/20 0.38
TSHR P16473 4/20 0.38
PDK2 Q15119 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAPT P10636 3/20 0.38
KDM4E B2RXH2 2/20 0.38
NFKB1 P19838 1/20 0.38
HTT P42858 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
TP53 P04637 1/20 0.37
POLB P06746 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29133127 1.00 BRD4 (0.47) BRD4NPC1RAB9ATDP1L3MBTL1
SCHEMBL30622243 0.78 BRD4 (0.36) BRD4NPC1RAB9ASMN1; SMN2POLB
SCHEMBL29133047 0.78 BRD4 (0.36) BRD4NPC1RAB9ASMN1; SMN2POLB
SCHEMBL29133096 0.78 RAB9A (0.44) BRD4NPC1RAB9AL3MBTL1SMN1; SMN2
SCHEMBL30622190 0.78 RAB9A (0.44) BRD4NPC1RAB9AL3MBTL1SMN1; SMN2
SCHEMBL4230324 0.76 NPC1 (0.65) BRD4NPC1RAB9ATDP1L3MBTL1
SCHEMBL8177826 0.75 RAB9A (0.47) BRD4NPC1RAB9ATDP1SMN1; SMN2
SCHEMBL4799665 0.72 IDO1 (0.37) KMT2AALDH1A1HPGDTSHRNPSR1
SCHEMBL15271912 0.71 BRD4 (0.41) BRD4NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL30622184 0.70 TDP1 (0.49) NPC1RAB9ATDP1L3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed