SCHEMBL30636331

SCHEMBL30636331

O=C(O)Cc1cccc2cnccc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.64
ROS1 P08922 1/20 0.58
RPS6KB1 P23443 1/20 0.58
GLS O94925 2/20 0.52
KDM4E B2RXH2 1/20 0.51
MAPKAPK2 P49137 1/20 0.51
MAPK8 P45983 10/20 0.50
MAPK10 P53779 10/20 0.50
MAPK9 P45984 9/20 0.50
CCNE1 P24864 1/20 0.49
CDK2 P24941 1/20 0.49
CDK5 Q00535 1/20 0.49
ALDH1A1 P00352 2/20 0.49
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
DAO P14920 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL837578 1.00 TDP1 (0.64) TDP1ROS1RPS6KB1GLSKDM4E
Hydrochloric Acid SCHEMBL3714409 0.98 TDP1 (0.62) TDP1ROS1RPS6KB1GLSKDM4E
SCHEMBL3714691 0.87 TDP1 (0.64) TDP1ROS1RPS6KB1GLSKDM4E
SCHEMBL3785081 0.85 ROS1 (0.56) ROS1RPS6KB1GLSKDM4EMAPKAPK2
SCHEMBL3721704 0.84 CCNC (0.52) TDP1ROS1RPS6KB1GLSKDM4E
SCHEMBL4022975 0.81 MAPK8 (0.58) TDP1ROS1RPS6KB1GLSMAPK8
Hydrochloric Acid SCHEMBL3941138 0.80 MAPK8 (0.57) TDP1ROS1RPS6KB1GLSMAPK8
SCHEMBL4022503 0.80 ROS1 (0.80) ROS1RPS6KB1GLSMAPK8MAPK10
SCHEMBL3711732 0.79 TDP1 (0.62) TDP1ROS1RPS6KB1KDM4EMAPK9
SCHEMBL30431204 0.79 TDP1 (0.62) TDP1ROS1RPS6KB1KDM4EMAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117062804-A 1, 3-substituted cyclobutyl derivatives and their use 诺华股份有限公司 2023-11-14 CN disclosed