SCHEMBL3721704

SCHEMBL3721704

O=C(O)CCc1cccc2cnccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.52
CDK8 P49336 1/20 0.52
ROS1 P08922 1/20 0.49
RPS6KB1 P23443 1/20 0.49
KDM4E B2RXH2 1/20 0.49
MAPKAPK2 P49137 1/20 0.49
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 1/20 0.47
GLS O94925 2/20 0.47
TRPV1 Q8NER1 2/20 0.46
SUCNR1 Q9BXA5 1/20 0.46
PARP1 P09874 1/20 0.46
DAO P14920 1/20 0.45
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30343669 0.88 CCNC (0.52) CCNCCDK8KDM4EMAPKAPK2KMT2A
SCHEMBL837578 0.84 TDP1 (0.64) ROS1RPS6KB1KDM4EMAPKAPK2KMT2A
SCHEMBL30636331 0.84 TDP1 (0.64) ROS1RPS6KB1KDM4EMAPKAPK2KMT2A
Hydrochloric Acid SCHEMBL3714409 0.83 TDP1 (0.62) ROS1RPS6KB1KDM4EMAPKAPK2KMT2A
SCHEMBL2849208 0.81 CCNC (0.48) CCNCCDK8KMT2APARP1CYP1A2
SCHEMBL30873960 0.81 CCNC (0.48) CCNCCDK8KMT2APARP1CYP1A2
SCHEMBL21350520 0.80 CCNC (0.52) CCNCCDK8ALDH1A1CYP1A2FFAR1
SCHEMBL6965122 0.80 CYP3A4 (0.50) ROS1RPS6KB1KDM4EMAPKAPK2KMT2A
SCHEMBL1830568 0.80 KDM4E (0.55) ROS1RPS6KB1KDM4EMAPKAPK2KMT2A
SCHEMBL30307853 0.80 TDP1 (0.67) KDM4EKMT2APARP1CYP1A2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010117090-A1 NOVEL ISOQUINOLINYLOXYMETHYL HETEROARYL DERIVATIVES BANYU PHARMACEUTICAL CO.,LTD. (JP) 2010-10-14 WO disclosed