SCHEMBL30641

SCHEMBL30641

O=C1c2cc(Br)ccc2CC12CCCC1=CCCC=C1C2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PARP1 P09874 1/20 0.35
PARP10 Q53GL7 1/20 0.35
TDP2 O95551 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA4 P22748 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
APP P05067 1/20 0.32
BACE1 P56817 1/20 0.32
PSMB5 P28074 1/20 0.32
TGM2 P21980 1/20 0.31
CES1 P23141 1/20 0.31
PDGFRB P09619 1/20 0.31
FGFR1 P11362 1/20 0.31
SRC P12931 1/20 0.31
KDR P35968 1/20 0.31
CMA1 P23946 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30859 0.87 TDP1 (0.41) TDP1L3MBTL1PARP1PARP10TDP2
SCHEMBL9948561 0.80 TDP1 (0.44) TDP1L3MBTL1PARP1PARP10TDP2
SCHEMBL1464516 0.80 L3MBTL1 (0.50) TDP1L3MBTL1PARP1PARP10APP
SCHEMBL1465245 0.78 L3MBTL1 (0.38) TDP1L3MBTL1PARP1PARP10TDP2
SCHEMBL9948162 0.77 TDP1 (0.46) TDP1L3MBTL1PARP1PARP10TDP2
SCHEMBL18087904 0.76 TDP1 (0.44) TDP1L3MBTL1PARP1PARP10TDP2
SCHEMBL7879908 0.76 TDP1 (0.35) TDP1L3MBTL1PARP1PARP10TGM2
SCHEMBL30642 0.76 TDP1 (0.35) TDP1L3MBTL1PARP1PARP10TGM2
SCHEMBL30482 0.75 TDP1 (0.45) TDP1L3MBTL1PARP1PARP10TDP2
SCHEMBL1465537 0.75 TDP1 (0.41) TDP1L3MBTL1PARP1PARP10TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406240-A2 INHIBITORS OF BETA-SECRETASE Vitae Pharmaceuticals, Inc. (US) 2012-01-18 EP disclosed
WO-2010105179-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-09-16 WO disclosed