Iofetamine

Iofetamine

SCHEMBL3064259

CC(C)N[C@H](C)Cc1ccc(I)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 1.00
CYP2D6 P10635 1/20 1.00
APEX1 P27695 1/20 0.96
PMP22 Q01453 1/20 0.96
SLC6A4 P31645 4/20 0.61
SIGMAR1 Q99720 5/20 0.50
TAAR1 Q96RJ0 2/20 0.41
SLC18A2 Q05940 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iofetamine SCHEMBL1534301 1.00 CYP1A2 (1.00) CYP1A2CYP2D6APEX1PMP22SLC6A4
Iofetamine SCHEMBL11151697 1.00 CYP1A2 (1.00) CYP1A2CYP2D6APEX1PMP22SLC6A4
Iofetamine SCHEMBL8973644 0.98 APEX1 (1.00) CYP1A2CYP2D6APEX1PMP22SLC6A4
Iofetamine SCHEMBL7755724 0.98 APEX1 (1.00) CYP1A2CYP2D6APEX1PMP22SLC6A4
Iofetamine SCHEMBL9860677 0.89 CYP1A2 (0.80) CYP1A2CYP2D6APEX1PMP22SLC6A4
Iofetamine SCHEMBL9860681 0.89 CYP1A2 (0.80) CYP1A2CYP2D6APEX1PMP22SLC6A4
SCHEMBL20862299 0.83 CYP1A2 (0.70) CYP1A2CYP2D6APEX1PMP22SLC6A4
SCHEMBL18211455 0.81 CYP1A2 (0.68) CYP1A2CYP2D6APEX1PMP22SLC6A4
SCHEMBL11265489 0.81 CYP2D6 (0.68) CYP1A2CYP2D6APEX1PMP22SLC6A4
SCHEMBL23986761 0.79 CYP1A2 (0.66) CYP1A2CYP2D6APEX1PMP22SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1004321-B1 STABLE RADIOACTIVE MEDECINE DAIICHI RADIOISOTOPE LAB (JP) 2003-02-26 EP claimed
EP-0485479-B1 PERFLUORO-T-BUTYL-CONTAINING COMPOUNDS FOR USE IN FLUORINE-19 NMR AND/OR MRI UNIV JOHNS HOPKINS (US) 1996-04-03 EP claimed
EP-0011858-B1 RADIOIODINE CONTAINING AMINES, THEIR PREPARATION AND THEIR USE AS BRAIN IMAGING AGENTS F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1983-05-18 EP claimed
CN-111393306-B Apparatus for synthesizing radioiodinated compound 日本医事物理股份有限公司 2021-03-26 CN disclosed
CN-111393306-A Apparatus for synthesizing radioiodinated compound 日本医事物理股份有限公司 2020-07-10 CN disclosed
US-9129373-B2 Apparatus for evaluating the accuracy of a SPECT or PET system using a phantom filled with a radioisotope NIHON MEDI-PHYSICS CO., LTD. (JP) 2015-09-08 US disclosed
US-20130251226-A1 APPARATUS FOR EVALUATING ACCURACY OF MEASUREMENT NATIONAL CEREBRAL AND CARDIOVASCULAR CENTER (JP) 2013-09-26 US disclosed
EP-1363954-B1 POLYMER PRECURSORS OF RADIOLABELED COMPOUNDS, AND METHODS OF MAKING AND USING THE SAME UNIV WESTERN ONTARIO (CA) 2012-10-17 EP disclosed
US-20100274052-A1 PREPARATION OF RADIOLABELLED HALOAROMATICS VIA POLYMER-BOUND INTERMEDIATES University of West Ontario 2010-10-28 US disclosed
US-7658910-B2 Preparation of radiolabelled haloaromatics via polymer-bound intermediates THE UNIVERSITY OF WESTERN ONTARIO (CA) 2010-02-09 US disclosed
EP-1197227-B9 METHOD OF THE ADMINISTRATION OF DRUGS HAVING BINDING AFFINITY WITH PLASMA PROTEIN AND PREPARATION TO BE USED IN THE METHOD NIHON MEDIPHYSICS CO LTD (JP) 2008-06-11 EP disclosed
EP-0335918-A1 DIAGNOSTIC OR RADIOTHERAPEUTIC COMPOSITION COMPRISING A HYDROGEN CONTAINING COMPOUND Mallinckrodt Diagnostica (Holland) B.V. (NL) 1989-10-11 EP disclosed
WO-1989001342-A2 DIAGNOSTIC OR RADIOTHERAPEUTIC COMPOSITION COMPRISING A HYDROGEN CONTAINING COMPOUND MALLINCKRODT, INC. (US) 1989-02-23 WO disclosed
US-4771059-A CENTRAL NERVOUS SYSTEM UNIVERSITY OF FLORIDA (US) 1988-09-13 US disclosed
EP-0174342-A1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES. UNIV FLORIDA (US) 1986-03-19 EP disclosed
EP-0165630-A2 Method of preparing a chlorinated, brominated, radiobrominated, iodinated and/or radioiodinated, aromatic or heteroaromatic compound, as well as a kit for preparing a diagnostic composition on the basis of this compound MALLINCKRODT, INC.(a Missouri corporation) (US) 1985-12-27 EP disclosed
WO-1985003937-A1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES UNIVERSITY OF FLORIDA (US) 1985-09-12 WO disclosed
EP-0011858-B1 RADIOIODINE CONTAINING AMINES, THEIR PREPARATION AND THEIR USE AS BRAIN IMAGING AGENTS F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1983-05-18 EP disclosed
US-4360511-A Amines useful as brain imaging agents MEDI-PHYSICS, INC. (US) 1982-11-23 US disclosed
EP-0011858-A1 Radioiodine containing amines, their preparation and their use as brain imaging agents F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1980-06-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100274052-A1 PREPARATION OF RADIOLABELLED HALOAROMATICS VIA POLYMER-BOUND INTERMEDIATES MPI, HDHD5, IPO5 CYP1A2 35/4885CYP2D6 212/4885APEX1 230/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.