SCHEMBL30644253

SCHEMBL30644253

Brc1ccc(N2CCN3CCOC[C@@H]3C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.47
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SOS1 Q07889 3/20 0.41
CYP1A1 P04798 1/20 0.40
CYP1B1 Q16678 1/20 0.40
MGLL Q99685 1/20 0.38
HSD17B10 Q99714 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
DPP4 P27487 1/20 0.36
CTSK P43235 3/20 0.35
CTSC P53634 3/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
PRCP P42785 1/20 0.35
L3MBTL3 Q96JM7 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
FGFR1 P11362 1/20 0.35
FGFR2 P21802 1/20 0.35
FGFR4 P22455 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31276654 1.00 AKR1C3 (0.47) AKR1C3MEN1KMT2ASOS1CYP1A1
SCHEMBL30644263 0.91 AKR1C3 (0.41) AKR1C3MEN1KMT2ASOS1CYP1A1
SCHEMBL16427192 0.85 AKR1C3 (0.49) AKR1C3MEN1KMT2ACYP1A1CYP1B1
SCHEMBL29964545 0.85 AKR1C3 (0.47) AKR1C3SOS1HRH3CTSKCTSC
SCHEMBL15551984 0.85 SOS1 (0.41) MEN1KMT2ASOS1HSD17B10HRH3
SCHEMBL29964729 0.85 AKR1C3 (0.47) AKR1C3SOS1HRH3CTSKCTSC
SCHEMBL29964783 0.85 AKR1C3 (0.47) AKR1C3SOS1HRH3CTSKCTSC
SCHEMBL16440196 0.85 AKR1C3 (0.47) AKR1C3MEN1KMT2ASOS1HSD17B10
SCHEMBL15551986 0.85 SOS1 (0.41) MEN1KMT2ASOS1HSD17B10HRH3
SCHEMBL16292255 0.82 AKR1C3 (0.49) AKR1C3MEN1KMT2ACYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117003755-A Pyrazolopyridazinone derivatives, compositions and uses thereof 北京伯汇生物技术有限公司 2023-11-07 CN disclosed