SCHEMBL30646115

SCHEMBL30646115

O=C1c2ccc(-c3cc(F)c(O)c(F)c3)nc2CCC1Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 7/20 0.47
CYP19A1 P11511 7/20 0.42
CYP24A1 Q07973 3/20 0.38
MAOB P27338 1/20 0.38
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
DHODH Q02127 1/20 0.35
HTR1A P08908 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
CYP27A1 Q02318 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30646096 0.85 MELK (0.35) CYP26A1CYP19A1CYP24A1DHODHCYP27A1
SCHEMBL30646127 0.82 CYP19A1 (0.37) CYP26A1CYP19A1DDB1CRBNDHODH
SCHEMBL30646108 0.79 MELK (0.34) DHODH
SCHEMBL4432336 0.73 CYP26A1 (0.38) CYP26A1CYP19A1CYP24A1DHODHCYP27A1
SCHEMBL30646131 0.68 GRM5 (0.44) DHODH
SCHEMBL8158688 0.67 CYP26A1 (0.86) CYP26A1CYP19A1CYP24A1HTR1ASIGMAR1
SCHEMBL8465475 0.65 CYP19A1 (0.78) CYP26A1CYP19A1CYP24A1HTR1ASIGMAR1
SCHEMBL4419499 0.64 CYP19A1 (0.38) CYP26A1CYP19A1CYP24A1DDB1CRBN
SCHEMBL4433213 0.64 CYP24A1 (0.43) CYP26A1CYP19A1CYP24A1MAOBDHODH
SCHEMBL3761876 0.63 CYP19A1 (0.80) CYP26A1CYP19A1MAOBDDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4543437-A1 3-?HSD1 INHIBITORS AND COMPOSITIONS AND USES THEREOF THE CLEVELAND CLINIC FOUNDATION (US) 2025-04-30 EP disclosed
WO-2023250480-A1 3-βHSD1 INHIBITORS AND COMPOSITIONS AND USES THEREOF THE CLEVELAND CLINIC FOUNDATION (US) 2023-12-28 WO disclosed