SCHEMBL30681963

SCHEMBL30681963

O=C(O)c1cccc(NC(=O)c2cc3cccnc3nc2N2CCCC(F)(F)CC2)c1

nearest known ligand 0.52

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KIF18A Q8NI77 3/20 0.52
SCN10A Q9Y5Y9 17/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26617813 1.00 KIF18A (0.52) KIF18ASCN10A
SCHEMBL26617951 0.92 SCN10A (0.53) KIF18ASCN10A
SCHEMBL30682007 0.92 SCN10A (0.53) KIF18ASCN10A
SCHEMBL30682013 0.91 SCN10A (0.51) KIF18ASCN10A
SCHEMBL26617559 0.91 SCN10A (0.51) KIF18ASCN10A
SCHEMBL30681997 0.91 SCN10A (0.51) KIF18ASCN10A
SCHEMBL30682040 0.86 KIF18A (0.60) KIF18ASCN10A
SCHEMBL30681897 0.86 SCN10A (0.50) KIF18ASCN10A
SCHEMBL30681930 0.86 SCN10A (0.68) KIF18ASCN10A
SCHEMBL26617815 0.86 SCN10A (0.68) KIF18ASCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119585247-A Bicyclic heterocyclic amide inhibitors of nav1.8 for the treatment of pain 赛特温治疗公司 2025-03-07 CN disclosed
EP-4514789-A1 <SUP2/>? <SUB2/>?V?BICYCLIC HETEROCYCLIC AMIDE INHIBITORS OF NA1.8 FOR THE TREATMENT OF PAIN SiteOne Therapeutics, Inc. (US) 2025-03-05 EP disclosed
WO-2023211990-A1 BICYCLIC HETEROCYCLIC AMIDE INHIBITORS OF NA V1.8 FOR THE TREATMENT OF PAIN SITEONE THERAPEUTICS, INC. (US) 2023-11-02 WO disclosed