SCHEMBL30686116

SCHEMBL30686116

C=CC[C@@H](C(=O)Cl)N(C)C(=O)O

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 2/20 0.32
GRIK2 Q13002 2/20 0.32
CYP2C19 P33261 1/20 0.32
CPA1 P15085 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27028742 1.00 GRIK1 (0.32) GRIK1GRIK2CYP2C19CPA1
SCHEMBL6674233 0.77 FAAH (0.32)
SCHEMBL29086756 0.73 GRIK1 (0.31) GRIK1GRIK2
SCHEMBL7164140 0.72 GRIK1 (0.39) GRIK1GRIK2CYP2C19CPA1
SCHEMBL466127 0.72 GRIK1 (0.39) GRIK1GRIK2CYP2C19CPA1
SCHEMBL6673351 0.72 GRIK1 (0.32) GRIK1GRIK2CYP2C19CPA1
SCHEMBL2973406 0.72 GRIK1 (0.36) GRIK1GRIK2CYP2C19CPA1
SCHEMBL2973400 0.72 GRIK1 (0.36) GRIK1GRIK2CYP2C19CPA1
SCHEMBL5764966 0.71 SLC6A2 (0.52)
Ammonia Solution, Strong SCHEMBL27395046 0.71 GRIK1 (0.38) GRIK1GRIK2CYP2C19CPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117279933-A Cyclic compounds having selective KRAS inhibition relative to HRAS and NRAS 中外制药株式会社 2023-12-22 CN disclosed