SCHEMBL30690908

SCHEMBL30690908

O=C(CCN1CCCCC1)N1CCN(c2ccc(F)cc2F)CC1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.54
DPP4 P27487 1/20 0.52
DPP9 Q86TI2 1/20 0.52
MAPT P10636 3/20 0.50
LMNA P02545 3/20 0.50
MEN1 O00255 1/20 0.50
TSHR P16473 1/20 0.50
KMT2A Q03164 1/20 0.50
ADRA1B P35368 2/20 0.49
ALDH1A1 P00352 2/20 0.49
HTR1A P08908 2/20 0.48
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48
HTR7 P34969 1/20 0.48
SIGMAR1 Q99720 2/20 0.47
PARP1 P09874 1/20 0.47
ACKR3 P25106 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
GPR174 Q9BXC1 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13419280 0.88 MAPT (0.50) MAPTLMNAMEN1TSHRKMT2A
SCHEMBL13419687 0.88 MAPT (0.48) DPP4DPP9MAPTLMNAMEN1
SCHEMBL3212037 0.84 DPP4 (0.56) DPP4MAPTLMNAMEN1KMT2A
SCHEMBL1903391 0.80 GRM5 (0.65) GRM5DPP4DPP9MAPTLMNA
SCHEMBL15840486 0.80 GRM5 (0.56) GRM5DPP4DPP9MAPTLMNA
SCHEMBL19002659 0.79 KMT2A (0.61) GRM5DPP4DPP9MAPTLMNA
SCHEMBL5659051 0.78 HTR1A (0.57) GRM5MAPTLMNAMEN1TSHR
SCHEMBL3796463 0.78 KMT2A (0.77) GRM5MAPTLMNAMEN1TSHR
SCHEMBL17208419 0.78 DPP4 (0.55) GRM5DPP4DPP9MAPTLMNA
SCHEMBL5655876 0.77 NOTUM (0.52) GRM5MAPTTSHRKMT2AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120443-A Compounds as adenosine A2a receptor antagonists and pharmaceutical compositions containing the same 株式会社 钟根堂 2023-11-24 CN disclosed