SCHEMBL30716245

SCHEMBL30716245

CC(C)c1cnn2c(NCc3ccccc3)nc(NC3CCC(C)(C)NC3)nc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 17/20 0.56
CDK9 P50750 15/20 0.56
CDK5 Q00535 4/20 0.55
CDK5R1 Q15078 4/20 0.55
CCNT1 O60563 2/20 0.55
CCNA2 P20248 2/20 0.55
DYRK3 O43781 1/20 0.55
CLK1 P49759 1/20 0.55
CLK2 P49760 1/20 0.55
CLK3 P49761 1/20 0.55
DYRK1A Q13627 1/20 0.55
DYRK2 Q92630 1/20 0.55
CLK4 Q9HAZ1 1/20 0.55
DYRK1B Q9Y463 1/20 0.55
CDK7 P50613 6/20 0.55
CCNH P51946 3/20 0.55
CCNE1 P24864 2/20 0.55
CDK4 P11802 2/20 0.53
MNAT1 P51948 2/20 0.46
CDK1 P06493 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30716232 0.87 CDK2 (0.49) CDK2CDK9CDK5CDK5R1CCNT1
SCHEMBL30716316 0.84 CDK7 (0.66) CDK2CDK9CDK7CCNHMNAT1
SCHEMBL30716320 0.80 CDK2 (0.45) CDK2CDK9CDK5CDK5R1CCNT1
SCHEMBL30716251 0.79 CDK2 (0.42) CDK2CDK9CDK5CDK5R1CCNT1
SCHEMBL26697016 0.77 CDK7 (0.42) CDK2CDK9CDK7CCNHCDK4
SCHEMBL30716295 0.76 CDK2 (0.41) CDK2CDK9CDK7CCNHCDK4
SCHEMBL31438142 0.75 CDK2 (0.70) CDK2CDK9CDK5CDK5R1CCNT1
SCHEMBL26341896 0.74 CDK2 (0.46) CDK2CDK9CDK5CDK5R1CCNT1
SCHEMBL26341883 0.74 CDK7 (0.47) CDK2CDK9CDK7CCNHCDK4
SCHEMBL26697001 0.73 CDK7 (0.51) CDK2CDK9CDK5CDK5R1CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023227125-A1 NEW FUSED-HETEROCYCLIC COMPOUND AS CDK INHIBITOR AND USE THEREOF 杭州德睿智药科技有限公司 2023-11-30 WO disclosed