SCHEMBL30716320

SCHEMBL30716320

CC(C)c1cnn2c(NCc3cc([N+](=O)[O-])ccc3Cl)nc(N[C@H]3CCC(C)(C)NC3)nc12

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 14/20 0.45
CDK9 P50750 14/20 0.45
CDK7 P50613 7/20 0.43
CDK4 P11802 2/20 0.43
CDK5 Q00535 2/20 0.40
CDK5R1 Q15078 2/20 0.40
DYRK3 O43781 1/20 0.40
CCNT1 O60563 1/20 0.40
CCNA2 P20248 1/20 0.40
CLK1 P49759 1/20 0.40
CLK2 P49760 1/20 0.40
CLK3 P49761 1/20 0.40
DYRK1A Q13627 1/20 0.40
DYRK2 Q92630 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
CCNH P51946 5/20 0.38
MNAT1 P51948 5/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30716232 0.87 CDK2 (0.49) CDK2CDK9CDK7CDK4CDK5
SCHEMBL26697019 0.81 CDK2 (0.42) CDK2CDK9CDK7CDK4CCNH
SCHEMBL26697025 0.81 CDK2 (0.42) CDK2CDK9CDK7CDK4CCNH
SCHEMBL30716295 0.81 CDK2 (0.41) CDK2CDK9CDK7CDK4CCNH
SCHEMBL30716245 0.80 CDK2 (0.56) CDK2CDK9CDK7CDK4CDK5
SCHEMBL26696894 0.77 CDK2 (0.39) CDK2CDK9CDK7CDK5CDK5R1
SCHEMBL30716316 0.73 CDK7 (0.66) CDK2CDK9CDK7CCNHMNAT1
SCHEMBL30716251 0.72 CDK2 (0.42) CDK2CDK9CDK7CDK4CDK5
SCHEMBL26697029 0.70 CDK9 (0.44) CDK2CDK9CDK7CDK4CCNH
SCHEMBL26697043 0.69 CDK7 (0.48) CDK2CDK9CDK7CDK4CCNH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023227125-A1 NEW FUSED-HETEROCYCLIC COMPOUND AS CDK INHIBITOR AND USE THEREOF 杭州德睿智药科技有限公司 2023-11-30 WO disclosed