SCHEMBL30716256

SCHEMBL30716256

C=CC(=O)Nc1cccc(Nc2nc(S(C)(=O)=O)nc3c(C(C)C)cnn23)c1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.48
CDK7 P50613 9/20 0.44
CCNH P51946 9/20 0.44
MNAT1 P51948 9/20 0.44
CSNK2A1 P68400 2/20 0.42
BTK Q06187 2/20 0.41
ITK Q08881 4/20 0.41
CDK2 P24941 1/20 0.40
CDK9 P50750 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26696916 1.00 EGFR (0.48) EGFRCDK7CCNHMNAT1CSNK2A1
SCHEMBL30716328 0.84 EGFR (0.49) EGFRCDK7CCNHMNAT1CSNK2A1
SCHEMBL26696830 0.84 EGFR (0.49) EGFRCDK7CCNHMNAT1CSNK2A1
SCHEMBL30716324 0.82 EGFR (0.52) EGFRCDK7CCNHMNAT1BTK
SCHEMBL19918771 0.82 CDK2 (0.43) CDK7CCNHMNAT1CSNK2A1CDK2
SCHEMBL30716274 0.81 CDK2 (0.45) CDK7CCNHCSNK2A1CDK2CDK9
SCHEMBL21473006 0.80 EGFR (0.45) EGFRCDK7CCNHMNAT1CSNK2A1
SCHEMBL18072717 0.79 CDK2 (0.41) EGFRCDK2CDK9
SCHEMBL21654892 0.78 CDK7 (0.56) EGFRCDK7CCNHMNAT1CSNK2A1
SCHEMBL18113858 0.75 CSNK2A1 (0.53) CDK7CCNHMNAT1CSNK2A1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023227125-A1 NEW FUSED-HETEROCYCLIC COMPOUND AS CDK INHIBITOR AND USE THEREOF 杭州德睿智药科技有限公司 2023-11-30 WO disclosed