SCHEMBL30718893

SCHEMBL30718893

CC(C)(C)CNc1nc(Cl)ncc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
NUDT1 P36639 3/20 0.44
MAPK8 P45983 4/20 0.41
MAPK9 P45984 1/20 0.41
MAPK10 P53779 1/20 0.41
STK17B O94768 2/20 0.36
STK17A Q9UEE5 2/20 0.36
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CTSL P07711 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
CDK1 P06493 2/20 0.34
CDK2 P24941 2/20 0.34
CCNB1 P14635 1/20 0.34
CCNE1 P24864 1/20 0.34
ABL1 P00519 1/20 0.33
BCR P11274 1/20 0.33
LRRK2 Q5S007 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4134213 1.00 MEN1 (0.46) MEN1KMT2ANUDT1MAPK8MAPK9
SCHEMBL1938007 0.83 STK17A (0.50) MEN1KMT2ANUDT1MAPK8STK17B
SCHEMBL13897499 0.81 MEN1 (0.52) MEN1KMT2ASTK17BSTK17AALDH1A1
SCHEMBL13649070 0.81 KMT2A (0.41) MEN1KMT2ASTK17BSTK17AALDH1A1
SCHEMBL4137651 0.80 NUDT1 (0.51) MEN1KMT2ANUDT1MAPK8MAPK9
SCHEMBL5436631 0.79 NUDT1 (0.43) MEN1KMT2ANUDT1MAPK8STK17B
SCHEMBL13649041 0.78 KMT2A (0.39) MEN1KMT2ASTK17BSTK17AALDH1A1
SCHEMBL3447092 0.78 KMT2A (0.50) MEN1KMT2ASTK17BSTK17AALDH1A1
SCHEMBL5786509 0.78 NUDT1 (0.45) MEN1KMT2ANUDT1MAPK8MAPK9
SCHEMBL5789412 0.78 NUDT1 (0.42) MEN1KMT2ANUDT1MAPK8MAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112469719-B Heterocondensed pyridone compounds and their use as IDH inhibitors 内尔维亚诺医疗科学公司 2024-01-23 CN disclosed