SCHEMBL30719998

SCHEMBL30719998

CCOC(=O)c1cc2cc(C(F)(F)F)cnc2n1[C@H](C)CNC(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.38
ADORA3 P0DMS8 2/20 0.36
ADORA2A P29274 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ABCB1 P08183 1/20 0.35
GAA P10253 2/20 0.35
ALDH1A1 P00352 2/20 0.35
CACNA1H O95180 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNA1C Q13936 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
RECQL P46063 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
ADORA1 P30542 1/20 0.34
AAK1 Q2M2I8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5222990 0.89 ADORA3 (0.38) ADORA3ADORA2AABCB1ALDH1A1MEN1
SCHEMBL5223742 0.87 BRD4 (0.37) ADORA3ADORA2AABCB1ADORA1AAK1
SCHEMBL5223751 0.87 BRD4 (0.37) ADORA3ADORA2AABCB1ADORA1AAK1
SCHEMBL29153689 0.83 POLB (0.43) POLBL3MBTL1GAAALDH1A1LMNA
SCHEMBL29153687 0.83 POLB (0.43) POLBL3MBTL1GAAALDH1A1LMNA
SCHEMBL5217792 0.82 ABCB1 (0.35) ADORA3ADORA2AABCB1LMNAADORA1
SCHEMBL5217784 0.82 ABCB1 (0.35) ADORA3ADORA2AABCB1LMNAADORA1
SCHEMBL5759888 0.82 PCSK9 (0.40) ADORA3ADORA2AL3MBTL1ABCB1ALDH1A1
SCHEMBL5759892 0.82 PCSK9 (0.40) ADORA3ADORA2AL3MBTL1ABCB1ALDH1A1
SCHEMBL5218644 0.82 BRD4 (0.37) ADORA3ADORA2AABCB1ADORA1AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396485-A PARP7 inhibitors 轩竹生物科技股份有限公司 2024-01-12 CN disclosed