SCHEMBL30728849

SCHEMBL30728849

OCn1ccc2c(-c3cn[nH]c3)ncnc21

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.46
PRMT5 O14744 1/20 0.38
SCN9A Q15858 1/20 0.36
TPH1 P17752 1/20 0.33
ADK P55263 1/20 0.33
PIK3CG P48736 1/20 0.33
AKT1 P31749 1/20 0.33
AKT2 P31751 1/20 0.33
P2RX7 Q99572 1/20 0.32
CHEK1 O14757 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30223679 0.87 SIGMAR1 (0.34) SIGMAR1TPH1
SCHEMBL13286173 0.86 SIGMAR1 (0.46) SIGMAR1PRMT5SCN9ATPH1PIK3CG
SCHEMBL21201777 0.80 SIGMAR1 (0.39) SIGMAR1PRMT5SCN9ATPH1
SCHEMBL10247590 0.80 SIGMAR1 (0.39) SIGMAR1PRMT5SCN9ATPH1PIK3CG
SCHEMBL24902073 0.79 SIGMAR1 (0.39) SIGMAR1PRMT5SCN9ATPH1P2RX7
SCHEMBL30749810 0.79 SIGMAR1 (0.39) SIGMAR1PRMT5SCN9ATPH1P2RX7
SCHEMBL871452 0.79 SIGMAR1 (0.39) SIGMAR1PRMT5SCN9ATPH1P2RX7
SCHEMBL13058244 0.79 SIGMAR1 (0.48) SIGMAR1PRMT5PIK3CGAKT1AKT2
SCHEMBL10222870 0.79 SIGMAR1 (0.45) SIGMAR1PRMT5PIK3CGAKT1AKT2
SCHEMBL13243498 0.79 SIGMAR1 (0.45) SIGMAR1PRMT5PIK3CGAKT1AKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117451899-A Method for detecting impurities in crude drug of amino acid protein kinase inhibitor 淄博高新技术产业开发区生物医药研究院 2024-01-26 CN claimed
CN-117451899-A Method for detecting impurities in crude drug of amino acid protein kinase inhibitor 淄博高新技术产业开发区生物医药研究院 2024-01-26 CN disclosed
CN-117451899-A Method for detecting impurities in crude drug of amino acid protein kinase inhibitor 淄博高新技术产业开发区生物医药研究院 2024-01-26 CN disclosed