SCHEMBL30729901

SCHEMBL30729901

O=[N+]([O-])c1ccc2c(cnn2Cc2cccc(F)c2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLS O94925 1/20 0.57
IDO1 P14902 1/20 0.52
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
EPHX2 P34913 2/20 0.48
PPARG P37231 2/20 0.48
EGFR P00533 7/20 0.46
ERBB2 P04626 7/20 0.46
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
MAPT P10636 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
SLC29A1 Q99808 1/20 0.42
CNR1 P21554 1/20 0.42
ACHE P22303 1/20 0.42
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL217553 1.00 GLS (0.57) GLSIDO1MEN1KMT2AEPHX2
SCHEMBL5435879 0.86 GLS (0.61) GLSKMT2ACYP1A2CYP2D6CYP2C19
SCHEMBL1728790 0.86 GLS (0.64) GLSMAPTCNR1ACHECNR2
SCHEMBL11002083 0.83 GLS (0.67) GLSMEN1KMT2AMAPTADORA2A
SCHEMBL3506368 0.83 GLS (0.54) GLSADORA2AADORA1RECQL
SCHEMBL3376313 0.83 GLS (0.54) GLSMEN1KMT2AEPHX2PPARG
SCHEMBL29377015 0.82 GLS (0.58) GLSEGFRERBB2GRIN1GRIN2B
SCHEMBL27083759 0.82 GLS (0.58) GLSEGFRERBB2GRIN1GRIN2B
SCHEMBL16213110 0.81 ERBB2 (0.61) MEN1KMT2AEGFRERBB2CYP1A2
SCHEMBL3378095 0.81 GLS (0.57) GLSGRIN1GRIN2BMAPTCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024026056-A2 HETEROARYL COMPOUNDS AS EGFR INHIBITORS AND THEIR USES ACCUTAR BIOTECHNOLOGY, INC. (US) 2024-02-01 WO disclosed