SCHEMBL30730798

SCHEMBL30730798

Nc1ncc(-c2cccc3nccn23)cc1-c1ccc(N2CCCC2=O)cn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 2/20 0.38
ROCK1 Q13464 2/20 0.38
CHEK1 O14757 1/20 0.38
MAP4K4 O95819 1/20 0.38
CSF1R P07333 1/20 0.38
PRKACA P17612 1/20 0.38
KDR P35968 1/20 0.38
MAP2K1 Q02750 1/20 0.38
ACVR1 Q04771 1/20 0.38
MAP4K2 Q12851 1/20 0.38
DYRK1A Q13627 1/20 0.38
AURKB Q96GD4 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
CNR2 P34972 1/20 0.36
ALOX5AP P20292 2/20 0.35
NR3C1 P04150 1/20 0.35
MAP4K1 Q92918 2/20 0.35
AKR1C3 P42330 1/20 0.35
HTR6 P50406 1/20 0.34
FEN1 P39748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22554214 1.00 CDK8 (0.38) CDK8ROCK1CHEK1MAP4K4CSF1R
SCHEMBL30731090 0.74 NPC1 (0.44) ALOX5APAKR1C3HTR6FEN1HRH3
SCHEMBL22554275 0.74 NPC1 (0.44) ALOX5APAKR1C3HTR6FEN1HRH3
SCHEMBL30731017 0.74 NPC1 (0.44) ALOX5APAKR1C3HTR6FEN1HRH3
SCHEMBL30730848 0.74 CNR2 (0.38) ACVR1CNR2ALOX5APAKR1C3HTR6
SCHEMBL22553813 0.74 CNR2 (0.38) ACVR1CNR2ALOX5APAKR1C3HTR6
SCHEMBL22553917 0.73 ALOX5AP (0.41) ACVR1CNR2ALOX5APAKR1C3FEN1
SCHEMBL30730773 0.73 ALOX5AP (0.41) ACVR1CNR2ALOX5APAKR1C3FEN1
SCHEMBL22553739 0.69 JAK2 (0.43) MAP4K4DYRK1ADYRK1BCNR2PIM1
SCHEMBL30730864 0.69 JAK2 (0.43) MAP4K4DYRK1ADYRK1BCNR2PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN claimed
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN disclosed