SCHEMBL30745169

SCHEMBL30745169

OCCc1ccc2ncc(Br)cc2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ALOX5 P09917 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
BACE1 P56817 1/20 0.39
PDE3B Q13370 2/20 0.37
PDE3A Q14432 2/20 0.37
P2RY12 Q9H244 2/20 0.37
CA2 P00918 1/20 0.34
CDK8 P49336 1/20 0.34
MAP4K4 O95819 1/20 0.34
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34
CDK1 P06493 1/20 0.34
KDR P35968 1/20 0.34
MET P08581 2/20 0.33
ACSS2 Q9NR19 1/20 0.33
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29151025 1.00 KDM4E (0.39) KDM4EALDH1A1ALOX5GAAMAPT
SCHEMBL2147979 0.86 HSD17B10 (0.37) CA2CDK8MAP4K4METNPC1
SCHEMBL30745166 0.85 PDGFRB (0.34) ALDH1A1MAPTBACE1METPDGFRB
SCHEMBL29151033 0.85 PDGFRB (0.34) ALDH1A1MAPTBACE1METPDGFRB
SCHEMBL14756190 0.83 TAAR1 (0.46) KDM4EALDH1A1GAAMAPTBACE1
SCHEMBL11154924 0.80 CYP1A2 (0.49) KDM4EALDH1A1ALOX5GAAMAPT
SCHEMBL14756200 0.80 TAAR1 (0.50) KDM4EALDH1A1MAPT
SCHEMBL31717019 0.79 DYRK1A (0.34) ALDH1A1MAPTBACE1METPDGFRB
SCHEMBL17242123 0.79 MALT1 (0.34) ALDH1A1MAPTBACE1METPDGFRB
SCHEMBL6519685 0.79 ROCK1 (0.41) BACE1CA2NPC1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117510470-A Pyridazinone compounds and application thereof 暨南大学 2024-02-06 CN disclosed