SCHEMBL30747006

SCHEMBL30747006

C[C@@]1(O)CCCN(c2ncnc3c(F)cncc23)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 2/20 0.39
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
JAK3 P52333 9/20 0.36
SIGMAR1 Q99720 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
PRKDC P78527 1/20 0.33
LCK P06239 1/20 0.33
NPC1 O15118 1/20 0.33
PKM P14618 1/20 0.33
LMNA P02545 1/20 0.33
PRNP P04156 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
PPARG P37231 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
NR2E3 Q9Y5X4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31553808 1.00 LRRK2 (0.39) LRRK2CCNCCDK8JAK3SIGMAR1
SCHEMBL30782481 0.84 ADORA3 (0.38) LRRK2JAK3PRKDCNPC1LMNA
SCHEMBL30961223 0.84 LRRK2 (0.39) LRRK2JAK3SCN10APRKDCLMNA
SCHEMBL30746978 0.84 LRRK2 (0.39) LRRK2JAK3SCN10APRKDCLMNA
SCHEMBL31553945 0.79 MAPT (0.50) CCNCCDK8JAK3SIGMAR1NPC1
SCHEMBL30746955 0.78 PRKDC (0.39) LRRK2CCNCCDK8JAK3SCN10A
SCHEMBL30746993 0.78 PRKDC (0.39) LRRK2CCNCCDK8JAK3SCN10A
SCHEMBL30883512 0.72 CYP1A2 (0.42) LRRK2SCN10A
SCHEMBL16190534 0.72 ACACB (0.46) LRRK2SIGMAR1ACACB
SCHEMBL31323088 0.72 PTK2 (0.49) LRRK2CCNCCDK8JAK3PRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117263959-A Preparation and application of aromatic KRAS mutant protein inhibitor 药雅科技(上海)有限公司 2023-12-22 CN disclosed