SCHEMBL3075427

SCHEMBL3075427

CC(C)(C)OC(=O)N[C@H]1CC[C@H](CCN2CCC(Oc3ccc(F)cc3C#N)CC2)CC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.56
DRD3 P35462 8/20 0.49
KCNA3 P22001 1/20 0.47
AAK1 Q2M2I8 1/20 0.45
HTR2A P28223 3/20 0.42
NSD2 O96028 1/20 0.42
HRH1 P35367 1/20 0.41
CCR3 P51677 1/20 0.41
KCNH2 Q12809 1/20 0.41
HTR1A P08908 1/20 0.41
DRD4 P21917 1/20 0.41
HTR2B P41595 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3963444 1.00 DRD2 (0.56) DRD2DRD3KCNA3AAK1HTR2A
SCHEMBL3067525 0.90 DRD3 (0.53) DRD2DRD3HTR2AHRH1CCR3
SCHEMBL3078178 0.90 DRD3 (0.53) DRD2DRD3HTR2AHRH1CCR3
SCHEMBL3075416 0.89 DRD2 (0.53) DRD2DRD3KCNA3HTR2AHRH1
SCHEMBL3962394 0.89 DRD2 (0.53) DRD2DRD3KCNA3HTR2AHRH1
SCHEMBL3082500 0.87 DRD3 (0.42) DRD2DRD3HTR2AHRH1CCR3
SCHEMBL3082496 0.87 DRD3 (0.42) DRD2DRD3HTR2AHRH1CCR3
SCHEMBL3083297 0.87 DRD3 (0.47) DRD2DRD3HTR2AHRH1CCR3
SCHEMBL3091198 0.87 DRD3 (0.47) DRD2DRD3HTR2AHRH1CCR3
SCHEMBL14715609 0.87 HRH1 (0.45) DRD2DRD3HTR2AHRH1CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7795437-B2 Ether derivatives HOFFMANN-LA ROCHE INC. (US) 2010-09-14 US disclosed