SCHEMBL30757382

SCHEMBL30757382

CCOCc1cc(C=O)ccc1-c1ccccc1S(=O)(=O)N(COC)c1noc(C)c1C

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 9/20 0.38
AGTR1 P30556 1/20 0.38
EDNRB P24530 2/20 0.33
ALDH1A1 P00352 1/20 0.32
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26688891 1.00 EDNRA (0.38) EDNRAAGTR1EDNRBALDH1A1RXFP1
SCHEMBL5529587 0.94 EDNRA (0.37) EDNRAAGTR1EDNRBALDH1A1
SCHEMBL30757333 0.94 EDNRA (0.37) EDNRAAGTR1EDNRBALDH1A1
SCHEMBL15728330 0.90 EDNRA (0.38) EDNRAAGTR1EDNRB
SCHEMBL5526164 0.90 EDNRA (0.34) EDNRAAGTR1ALDH1A1RXFP1
SCHEMBL26688997 0.89 NPC1 (0.36) EDNRAAGTR1EDNRBALDH1A1
SCHEMBL30757507 0.89 NPC1 (0.36) EDNRAAGTR1EDNRBALDH1A1
SCHEMBL30517192 0.89 EDNRA (0.38) EDNRAAGTR1EDNRBALDH1A1
SCHEMBL30757240 0.87 EDNRA (0.43) EDNRAAGTR1EDNRB
SCHEMBL535104 0.87 EDNRA (0.43) EDNRAAGTR1EDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023224963-A1 DUAL-ACTING ANGIOTENSIN AND ENDOTHELIN RECEPTOR ANTAGONISTS ARIA PHARMACEUTICALS, INC. (US) 2023-11-23 WO disclosed