SCHEMBL30768115

SCHEMBL30768115

CSc1ncc2cc(C(F)F)nc(Cl)c2n1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HASPIN Q8TF76 2/20 0.39
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.30
HTT P42858 1/20 0.30
PIM1 P11309 1/20 0.30
TTK P33981 1/20 0.30
PIM2 Q9P1W9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26341306 1.00 HASPIN (0.39) HASPINMEN1KMT2AALDH1A1GAA
SCHEMBL20203577 0.81 HASPIN (0.36) HASPINMEN1KMT2AGAAHTT
SCHEMBL30460896 0.79 KMT2A (0.44) HASPINMEN1KMT2AALDH1A1GAA
SCHEMBL25275333 0.79 KMT2A (0.44) HASPINMEN1KMT2AALDH1A1GAA
SCHEMBL27034848 0.78 HASPIN (0.42) HASPINMEN1KMT2AALDH1A1GAA
SCHEMBL15507768 0.78 HASPIN (0.42) HASPINMEN1KMT2AALDH1A1GAA
SCHEMBL20037627 0.77 HASPIN (0.36) HASPINPIM1TTKPIM2
SCHEMBL26181506 0.76 HASPIN (0.35) HASPIN
SCHEMBL30460946 0.76 HASPIN (0.39) HASPINMEN1KMT2AALDH1A1GAA
SCHEMBL25230364 0.76 HASPIN (0.39) HASPINMEN1KMT2AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4558502-A1 AZA-QUINAZOLINE COMPOUNDS AND METHODS OF USE Iambic Therapeutics, Inc. (US) 2025-05-28 EP disclosed
CN-120051470-A Azaquinazoline compounds and methods of use 依安彼克医疗有限公司 2025-05-27 CN disclosed
WO-2024020419-A1 AZA-QUINAZOLINE COMPOUNDS AND METHODS OF USE IAMBIC THERAPEUTICS, INC. (US) 2024-01-25 WO disclosed