SCHEMBL30768149

SCHEMBL30768149

O=[N+]([O-])c1ccc(N2CCc3c(Br)cccc3C2)cc1

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.67
KMT2A Q03164 3/20 0.67
SIRT6 Q8N6T7 2/20 0.48
MAPT P10636 6/20 0.47
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 2/20 0.44
POLB P06746 1/20 0.44
ADRB1 P08588 1/20 0.44
LMNA P02545 1/20 0.44
APOBEC3G Q9HC16 1/20 0.43
GAA P10253 1/20 0.42
ABHD6 Q9BV23 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29201123 1.00 MEN1 (0.67) MEN1KMT2ASIRT6MAPTKDM4E
SCHEMBL6609282 0.80 MEN1 (1.00) MEN1KMT2ASIRT6MAPTKDM4E
SCHEMBL28457709 0.80 EED (0.46) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL28940436 0.79 ACACB (0.56) MAPTKDM4EALDH1A1LMNA
SCHEMBL29644378 0.79 ACACB (0.56) MAPTKDM4EALDH1A1LMNA
SCHEMBL28739023 0.78 HPGD (0.70) MEN1KMT2AMAPTALDH1A1POLB
SCHEMBL29644426 0.78 HPGD (0.70) MEN1KMT2AMAPTALDH1A1POLB
SCHEMBL30874289 0.76 HTR3E (0.42) MEN1KMT2AMAPTKDM4EALDH1A1
SCHEMBL29229997 0.76 HTR3E (0.42) MEN1KMT2AMAPTKDM4EALDH1A1
SCHEMBL7995398 0.72 KMT2A (0.65) MEN1KMT2ASIRT6MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114507181-B Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-03-26 CN disclosed