SCHEMBL307703

SCHEMBL307703

COc1ccc(C(=O)Nc2cccc(C(=O)Nc3ccc4c(c3)CN(Cc3ccc(F)cc3F)CC4)c2)cc1OC

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.57
CYP3A4 P08684 1/20 0.57
ABCG2 Q9UNQ0 5/20 0.53
ABCB1 P08183 4/20 0.53
ALDH1A1 P00352 1/20 0.49
POLB P06746 1/20 0.49
GAA P10253 1/20 0.49
NPC1 O15118 1/20 0.48
DRD2 P14416 1/20 0.48
DRD3 P35462 1/20 0.48
PRKG1 Q13976 1/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 1/20 0.47
TNF P01375 1/20 0.47
RAB9A P51151 1/20 0.47
NOD2 Q9HC29 1/20 0.47
NOD1 Q9Y239 1/20 0.47
ATM Q13315 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL306999 0.92 ROCK2 (0.71) ROCK2CYP3A4ABCG2ABCB1DRD2
SCHEMBL306402 0.89 ROCK2 (0.58) ROCK2CYP3A4ABCG2ABCB1ALDH1A1
SCHEMBL308954 0.88 ROCK2 (0.62) ROCK2CYP3A4ABCG2ABCB1ALDH1A1
SCHEMBL307835 0.84 ROCK2 (0.73) ROCK2CYP3A4ABCG2ABCB1DRD2
SCHEMBL307753 0.82 ROCK2 (0.75) ROCK2CYP3A4ABCG2ABCB1DRD2
SCHEMBL307225 0.82 ROCK2 (0.75) ROCK2CYP3A4ABCG2ABCB1PRKG1
SCHEMBL306148 0.82 ROCK2 (0.72) ROCK2CYP3A4ABCG2ABCB1DRD2
SCHEMBL307344 0.80 ROCK2 (0.75) ROCK2CYP3A4ABCG2ABCB1PRKG1
SCHEMBL307750 0.80 ROCK2 (0.75) ROCK2CYP3A4ABCG2ABCB1PRKG1
SCHEMBL14135092 0.78 ROCK2 (0.74) ROCK2CYP3A4ABCG2ABCB1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093266-B2 Rho kinase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-10 US claimed