Terikalant

Terikalant

SCHEMBL30770792

COc1ccc(C2CCN(CC[C@H]3CCOc4ccccc43)CC2)cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 1.00
DRD2 P14416 3/20 0.44
NPSR1 Q6W5P4 1/20 0.42
SLC6A4 P31645 1/20 0.41
TLR9 Q9NR96 3/20 0.41
TLR7 Q9NYK1 3/20 0.41
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
ABCB1 P08183 1/20 0.40
TLR4 O00206 1/20 0.40
TLR3 O15455 1/20 0.40
TLR8 Q9NR97 1/20 0.40
HTR2A P28223 1/20 0.40
QDPR P09417 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Terikalant SCHEMBL1815992 1.00 KCNH2 (1.00) KCNH2DRD2NPSR1SLC6A4TLR9
Terikalant SCHEMBL9678648 1.00 KCNH2 (1.00) KCNH2DRD2NPSR1SLC6A4TLR9
Terikalant SCHEMBL9772825 0.99 KCNH2 (0.98) KCNH2DRD2NPSR1SLC6A4TLR9
SCHEMBL18509377 0.94 KCNH2 (0.89) KCNH2DRD2ABCB1
SCHEMBL9014359 0.94 KCNH2 (0.89) KCNH2DRD2NPSR1TLR9TLR7
Terikalant SCHEMBL10407782 0.92 KCNH2 (0.84) KCNH2DRD2ACHEHTR2A
Terikalant SCHEMBL1230246 0.92 KCNH2 (0.84) KCNH2DRD2ACHEHTR2A
Terikalant SCHEMBL1230245 0.92 KCNH2 (0.84) KCNH2DRD2ACHEHTR2A
Terikalant SCHEMBL10407783 0.92 KCNH2 (0.84) KCNH2DRD2ACHEHTR2A
SCHEMBL10407769 0.91 KCNH2 (0.84) KCNH2DRD2QDPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024091485-A1 COMPOSITIONS AND METHODS FOR TREATING OR PREVENTING PULMONARY FIBROSIS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-05-02 WO disclosed
EP-3355925-B1 TREATMENT OF ACUTE TRAUMATIC INJURY UNIV ROCHESTER (US) 2024-02-28 EP disclosed