SCHEMBL307708

SCHEMBL307708

COc1ccc(C(=O)Nc2cccc(C(=O)Nc3nc4c(s3)CN(CCF)CC4)c2)cc1OC

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 13/20 0.61
NPC1 O15118 2/20 0.56
CYP1A2 P05177 2/20 0.56
CYP2C19 P33261 2/20 0.56
RAB9A P51151 2/20 0.56
CYP2D6 P10635 1/20 0.56
HPGD P15428 1/20 0.56
GAA P10253 1/20 0.54
KDM4E B2RXH2 1/20 0.52
ROCK1 Q13464 1/20 0.51
TP53 P04637 2/20 0.50
MAPT P10636 2/20 0.50
MEN1 O00255 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CASP1 P29466 1/20 0.50
CASP7 P55210 1/20 0.50
KMT2A Q03164 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ALOX15 P16050 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL306647 0.89 ROCK2 (0.65) ROCK2ROCK1CYP3A4
SCHEMBL308100 0.82 ROCK2 (0.66) ROCK2ROCK1CYP3A4
SCHEMBL307655 0.81 ROCK2 (0.63) ROCK2ROCK1CYP3A4
SCHEMBL307660 0.79 ROCK2 (0.62) ROCK2ROCK1CYP3A4
SCHEMBL307404 0.79 ROCK2 (0.64) ROCK2NPC1CYP2C19RAB9AGAA
SCHEMBL307096 0.78 ROCK2 (0.78) ROCK2NPC1CYP1A2CYP2C19RAB9A
SCHEMBL10311072 0.76 ROCK2 (1.00) ROCK2NPC1CYP1A2CYP2C19RAB9A
SCHEMBL10311071 0.76 ROCK2 (1.00) ROCK2NPC1CYP1A2CYP2C19RAB9A
SCHEMBL306952 0.74 ROCK2 (0.65) ROCK2NPC1CYP1A2CYP2C19RAB9A
SCHEMBL10070399 0.73 ROCK2 (0.79) ROCK2NPC1CYP1A2CYP2C19RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093266-B2 Rho kinase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-10 US claimed