SCHEMBL30775154

SCHEMBL30775154

CC(C)(C)[Si](C)(C)Oc1ccc(C2(O)CN(c3cc(C(=O)O)ccn3)C2)c(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 14/20 0.54
HSD17B13 Q7Z5P4 1/20 0.54
PIK3CA P42336 1/20 0.42
KDM5A P29375 5/20 0.38
KDM5B Q9UGL1 5/20 0.38
KDM4C Q9H3R0 4/20 0.38
KDM4A O75164 1/20 0.36
KDM2B Q8NHM5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29216000 1.00 NR1H4 (0.54) NR1H4HSD17B13PIK3CAKDM5AKDM5B
SCHEMBL19202590 0.91 NR1H4 (0.46) NR1H4HSD17B13PIK3CAKDM5AKDM5B
SCHEMBL19689544 0.83 NR1H4 (0.39) NR1H4HSD17B13
SCHEMBL30064297 0.83 NR1H4 (0.39) NR1H4HSD17B13
SCHEMBL17843256 0.82 PIK3CA (0.39) NR1H4HSD17B13PIK3CAKDM5AKDM5B
SCHEMBL29139872 0.80 NR1H4 (0.53) NR1H4HSD17B13PIK3CAKDM5AKDM5B
SCHEMBL30775159 0.80 NR1H4 (0.53) NR1H4HSD17B13PIK3CAKDM5AKDM5B
SCHEMBL22320341 0.80 CA12 (0.39) NR1H4HSD17B13
SCHEMBL20749493 0.77 NR1H4 (0.49) NR1H4HSD17B13PIK3CAKDM5AKDM5B
Nitrous Acid SCHEMBL29139870 0.76 NR1H4 (0.51) NR1H4HSD17B13PIK3CAKDM5AKDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117924266-A Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-04-26 CN disclosed
CN-117924267-A Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-04-26 CN disclosed
CN-109476636-B Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-01-09 CN disclosed