SCHEMBL19202590

SCHEMBL19202590

COC(=O)c1ccnc(N2CC(O)(c3ccc(O[Si](C)(C)C(C)(C)C)cc3Cl)C2)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 10/20 0.46
HSD17B13 Q7Z5P4 1/20 0.46
KDM5A P29375 4/20 0.38
KDM5B Q9UGL1 4/20 0.38
HRH3 Q9Y5N1 2/20 0.36
PIK3CA P42336 1/20 0.36
KDM4C Q9H3R0 2/20 0.34
KDM4E B2RXH2 2/20 0.34
ALOX15 P16050 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ACLY P53396 1/20 0.34
KDM6B O15054 1/20 0.33
KDM5C P41229 1/20 0.33
KDM2A Q9Y2K7 1/20 0.33
KDM3A Q9Y4C1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17843256 0.91 PIK3CA (0.39) NR1H4HSD17B13KDM5AKDM5BHRH3
SCHEMBL29216000 0.91 NR1H4 (0.54) NR1H4HSD17B13KDM5AKDM5BPIK3CA
SCHEMBL30775154 0.91 NR1H4 (0.54) NR1H4HSD17B13KDM5AKDM5BPIK3CA
SCHEMBL19202591 0.83 NR1H4 (0.45) NR1H4HSD17B13KDM5AKDM5BHRH3
SCHEMBL30064297 0.81 NR1H4 (0.39) NR1H4HSD17B13HRH3
SCHEMBL19689544 0.81 NR1H4 (0.39) NR1H4HSD17B13HRH3
SCHEMBL30775168 0.81 NR1H4 (0.51) NR1H4
SCHEMBL19689515 0.81 NR1H4 (0.51) NR1H4
SCHEMBL22320341 0.76 CA12 (0.39) NR1H4HSD17B13
SCHEMBL19202535 0.76 NR1H4 (0.44) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017128896-A1 FXR AGONIST AND PREPARATION METHOD AND USE THEREOF 江苏豪森药业集团有限公司 2017-08-03 WO disclosed