SCHEMBL30775162

SCHEMBL30775162

COC(=O)c1cnc(N2CC(O)(c3ccc(O)cc3Cl)C2)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 11/20 0.51
P2RY12 Q9H244 4/20 0.41
ABL1 P00519 1/20 0.37
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
OPRK1 P41145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19689507 1.00 NR1H4 (0.51) NR1H4P2RY12ABL1HDAC3HDAC1
SCHEMBL19689515 0.84 NR1H4 (0.51) NR1H4P2RY12ABL1
SCHEMBL30775168 0.84 NR1H4 (0.51) NR1H4P2RY12ABL1
SCHEMBL19699381 0.82 NR1H4 (0.46) NR1H4HDAC3HDAC1HDAC2HDAC6
SCHEMBL19202591 0.78 NR1H4 (0.45) NR1H4
SCHEMBL17843228 0.77 CRBN (0.52) NR1H4P2RY12
SCHEMBL19690321 0.77 NR1H4 (0.40) NR1H4
SCHEMBL30775163 0.76 NR1H4 (0.77) NR1H4
SCHEMBL19689549 0.76 NR1H4 (0.77) NR1H4
SCHEMBL19689491 0.75 NR1H4 (0.86) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117924266-A Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-04-26 CN disclosed
CN-117924267-A Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-04-26 CN disclosed
CN-109476636-B Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-01-09 CN disclosed